Acetylcholine Muscarinic Receptors



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Catalog No. Product Name Application Product Information
A11166

5-hydroxymethyl tolterodine (PNU 200577)

muscarinic receptor antagonist

5-hydroxymethyl tolterodine is a metabolite of Tolterodine, a muscarinic receptor antagonist used in the treatment of urinary incontinence.

A10032

Acetylcysteine

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Acetylcysteine is a pharmaceutical drug and nutritional supplement used primarily as a mucolytic agent and in the management of paracetamol (acetaminophen) overdose. Oral acetylcysteine is also used for the prevention of radiocontrast-induced nephropathy (a form of acute renal failure).

A13071

Arecoline

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Arecoline is a cholinergic alkaloid from seeds of the betel nut palm Areca catechu.
A10098

Atropine

AChR antagonist
Atropine is a competitive antagonist for the muscarinic acetylcholine receptor types M1, M2, M3, M4 and M5.
A10180

Bethanechol chloride

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Bethanechol is a parasympathomimetic choline carbamate that selectively stimulates muscarinic receptors without any effect on nicotinic receptors.
A10147

Biperiden HCl

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Biperiden hydrochloride is a muscarinic receptor antagonist that displays some selectivity for the M1 subtype
A11987

Darifenacin

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Darifenacin works by blocking the M3 muscarinic acetylcholine receptor, which is primarily responsible for bladder muscle contractions.
A10386

Fesoterodine fumarate (Toviaz)

AChR antagonist
Fesoterodine fumarate is a medicine which is used in urinary urgency, reducing the frequency of passing urine and urge urinary incontinence
A10416

Galanthamine hydrobromide

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Galanthamine is an AChE inhibitor with IC50 of 14 nM.
A10417

Gallamine triethiodide

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Gallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity.
A10476

Ipratropium bromide

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Ipratropium bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine.
A10480

Irsogladine

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Rsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.
A11975

Methoctramine hydrate

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Methoctramine hydrate is a selective M2 muscarinic receptor antagonist at nM concentrations
A10579

Methscopolamine bromide

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Methscopolamine bromide is a competitive antimuscarinic agent that blocks the binding of acetylcholine at muscarinic acetylcholine receptors (mAChR M).
A10635

Neostigmine bromide (Prostigmin)

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Neostigmine bromide is a reversible acetylcholine esterase inhibitor that binds to the anionic binding site of AChE.
A11712

Orphenadrine citrate

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Orphenadrine is known to have the following pharmacology: mACh receptor antagonist (anticholinergic); H1 receptor antagonist (antihistamine); NMDA receptor antagonist; NET blocker (norepinephrine reuptake inhibitor); Nav1.7, Nav1.8, and Nav1.9 sodium channel blocker; HERG potassium channel blocker.
A10684

Oxybutynin

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Oxybutynin(Ditropan) is an anticholinergic medication used to relieve urinary and bladder difficulties.
A11719

Rivastigmine tartrate

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Rivastigmine tartrate is a dual cholinesterase inhibitor (ChEI). It inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE).
A10803

Rocuronium bromide

TGF-βR inhibitor
Rocuronium bromide is an aminosteroid non-depolarizing neuromuscular blocker and also is used as a muscle relaxant used in modern anesthesia to facilitate endotracheal intubation.
A11215

Solifenacin succinate

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Solifenacin-succinate is a muscarinic M3 receptor antagoinst, used in treatment of urinary incontinence.
A10808

SVT-40776 (Tarafenacin)

muscarinic receptor antagonist
SVT-40776 is a novel M3 muscarinic receptor antagonist, for the treatment of overactive bladder.
A10937

Tolterodine tartrate (Detrol LA)

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Tolterodine tartrate (Detrol LA) is a muscarinic receptor antagonist which is used for the treatment of urinary incontinence.
A11706

Tropicamide

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Tropicamide is an anticholinergic used as a mydriatic.

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