AChR



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Catalog No. Product Name Application Product Information
A13761

(-)-Nicotine ditartrate

-
(-)-Nicotine ditartrate is a potent agonist of AChR (nicotinic acetylcholine recepto).
A11166 SALE

5-hydroxymethyl tolterodine (PNU 200577)

muscarinic receptor antagonist

5-hydroxymethyl tolterodine is a metabolite of Tolterodine, a muscarinic receptor antagonist used in the treatment of urinary incontinence.

A13539

A-582941

α7 nAChR agonist
A-582941 is a selective AChR a7 partial agonist. It exhibits high affinity for both rat and human a7 receptors (Ki values are 10.8 and 16.7 nM, respectively).
A11290

A-867744

modulator of α7 nAChRs
A-867744 is a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.
A16390

Acetylcholine iodide

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Acetylcholine iodide is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the central nervous system.
A15782

Acotiamide hydrochloride trihydrate

Acetylcholinesterase inhibitor
Acotiamide is a drug approved in Japan for the treatment of postprandial fullness, upper abdominal bloating, and early satiation due to functional dyspepsia.
A13071 SALE

Arecoline

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Arecoline is a cholinergic alkaloid from seeds of the betel nut palm Areca catechu.
A10098

Atropine

AChR antagonist
Atropine is a competitive antagonist for the muscarinic acetylcholine receptor types M1, M2, M3, M4 and M5.
A13653

Benzethonium Chloride

nAChR inhibitor
Benzethonium chloride is a potent inhibitor of nAChRs, it inhibits α4β2 nAChRs and α7 nAChRs with IC50 of 49 nM and 122 nM, respectively.
A10180 SALE

Bethanechol chloride

Muscarinic receptor agonist
Bethanechol is a parasympathomimetic choline carbamate that selectively stimulates muscarinic receptors without any effect on nicotinic receptors.
A10147 SALE

Biperiden HCl

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Biperiden hydrochloride is a muscarinic receptor antagonist that displays some selectivity for the M1 subtype
A12161

Catharanthine sulfate

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Catharanthine sulfate is a vinblastine-type alkaloid precursor with antitumor activity. It inhibits AChR by ion channel blocking and desensitization.
A11987

Darifenacin

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Darifenacin works by blocking the M3 muscarinic acetylcholine receptor, which is primarily responsible for bladder muscle contractions.
A13925

Deoxyvasicine HCl

AChE inhibitor
Desoxypeganine hydrochloride is an AChE (acetylcholinesterase) inhibitor that has been used in the treatment of Alzheimer's dementia.
A10330 SALE

Donepezil hydrochloride

cholinesterase inhibitor
Donepezil is a centrally acting reversible acetylcholinesterase inhibitor.
A15086

EVP-6124

nAChR Inhibitor
EVP-6124 is a novel partial agonist of ??7 neuronal nicotinic acetylcholine receptors (nAChRs); shows selectivity for ??7 nAChRs and did not activate or inhibit heteromeric ??4??2 nAChRs.
A15087

EVP-6124 hydrochloride

nAChR Inhibitor
EVP-6124 hydrochloride is a novel partial agonist of ??7 neuronal nicotinic acetylcholine receptors (nAChRs). EVP-6124 showed selectivity for ??7 nAChRs and did not activate or inhibit heteromeric ??4??2 nAChRs.
A10386 SALE

Fesoterodine fumarate (Toviaz)

AChR antagonist
Fesoterodine fumarate is a medicine which is used in urinary urgency, reducing the frequency of passing urine and urge urinary incontinence
A12900 SALE

Flavoxate

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Flavoxate binds and inhibits muscarinic receptors, thereby suppressing the micturition reflex and increases urinary bladder capacity by modifying the micturition center in the brain stem.
A10416 SALE

Galanthamine hydrobromide

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Galanthamine is an AChE inhibitor with IC50 of 14 nM.
A10417 SALE

Gallamine triethiodide

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Gallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity.
A12641

Glycopyrrolate

muscarinic antagonist
Glycopyrrolate is a muscarinic competitive antagonist used as an antispasmodic.
A15950

GTS-21 (DMBX-A)

nAChR agonist
GTS-21 dihydrochloride is a selective α7 nicotinic acetylcholine receptor agonist, has recently been established as a promising treatment for inflammation.
A10476

Ipratropium bromide

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Ipratropium bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine.
A10480 SALE

Irsogladine

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Rsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.

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