Cathepsin

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  1. Inhibitor (18)


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Catalog No. Product Name Application Product Information
A15290

Acetyl-Calpastatin (184-210) (human)

Selective calpain inhibitor
Acetyl-Calpastatin (184-210) (human), selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 uM). Increases secretion of amyoid ??-protein (A??) 42, A??40 and A??42 ratio.
A12020

Balicatib

Cathepsin K inhibitor
Balicatib, a cathepsin K inhibitor, stimulates periosteal bone formation in monkeys.
A13256

CA-074

Cathepsin B inhibitor
A14911

Calpain Inhibitor II, ALLM

Calpain Inhibitor
Calpain Inhibitor II, ALLM is a cell-permeable inhibitor of calpain I, calpain II, cathepsin L and cathepsin B with Ki values of 120 nM, 230 nM, 0.6 nM and 100 nM, respectively.
A15295

Calpeptin

Calpain inhibitor
Calpeptin is a cell permeable calpain inhibitor.
A11466

Cathepsin Inhibitor 1

Cathepsin Inhibitor
Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.
A13259

E 64d (Aloxistatin)

Cysteine Protease inhibitor
E-64d is an inhibitor of cathepsins B and L and it is lysosome and cell permeable.
A13257

E-64

Cysteine Protease inhibitor
E-64 is an irreversible and selective cysteine protease inhibitor with IC50 of 9 nM for papain.
A14145

Leupeptin hemisulfate

Cysteine Protease inhibitor
Leupeptin hemisulfate is a reversible inhibitor of trypsin-like and cysteine proteases such as calpain.
A13258

Loxistatin Acid (E64-C)

Cysteine Protease inhibitor
Loxistatin Acid, a derivative of E-64, is an irreversible and membrane-permeant cysteine protease inhibitor.
A15303

MDL 28170

Calpain Inhibitor III
MDL 28170 is a cell permeable selective inhibitor of Calpain 1, a Ca2+-dependent cysteine protease which has been implicated in apoptosis of immune cells as well as neuronal cells.
A14220

MG-101

Cysteine Protease inhibitor
MG-101 (ALLN) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.
A11265

Odanacatib (MK-0822)

Cathepsin K Inhibitor
Odanacatib is an inhibitor of cathepsin K,an enzyme involved in bone resorption.
A15306

PD 150606

Non-peptide calpain inhibitor
PD 150606 is a cell-permeable, non-competitive, selective, non-peptide Ca2+ dependent calpain inhibitor for calpain-1 and for calpain-2 directed towards the Ca2+ binding sites of calpain.
A14245

PD 151746

Calpain inhibitor
PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain.
A11901

PMSF

Serine/cysteine protease inhibitor
PMSF is an irreversible serine/cysteine protease inhibitor.
A13640

SJA6017

reversible Calpain inhibitor
SJA6017 is a cell permeable peptide aldehyde which functions as a reversible calpain inhibitor.
A14284

Z-FA-FMK

Irreversible Cysteine Protease inhibitor
Z-FA-FMK is an irreversible cysteine protease inhibitor.

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