CGRP Receptor

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  1. CGRP Receptor antagonist

    MK 3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.
  2. CGRP receptor antagonist

    MK-0974 (Telcagepant) is a potent and selective antagonist of the human and rhesus CGRP receptors.
  3. CGRP1 receptor

    Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.
  4. CGRP receptor antagonist

    BMS-927711 is a potent, selective, competitive human calcitonin gene-related peptide (CGRP) receptor antagonist that has shown in vivo efficacy without vasoconstrictor effect.
  5. CGRP Receptor antagonist

    MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3.
  6. CGRP receptor antagonist

    HCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor.

  7. CGRP antagonist

    Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine.
  8. CGRP1 receptor antagonist

    Olcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.

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