TG100-115Catalog No. A10922

Quick Overview

TG100-115 inhibits PI3K γ and -δ(IC50 values of 83 and 235 nM, respectively).
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TG100-115

Product Information
Catalog Num A10922
M. Wt 346.3
Formula C18H14N6O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 677297-51-7
Synonyms TG100115
Chemical Name 3-[2,4-diamino-6-(3-hydroxyphenyl)pteridin-7-yl]phenol (6,7-Bis(3-hydroxyphenyl)pteridine-2,4-diamine)
SMILES Code C1=CC(=CC(=C1)O)C2=NC3=C(N=C2C4=CC(=CC=C4)O)N=C(N=C3N)N

Biological activity
Introduction
TG100-115 inhibits PI3K γ and -δ(IC50 values of 83 and 235 nM, respectively).
Targets
PI3Kγ PI3Kδ PI3Kβ PI3Kα
83 nM235 nM1.2 μM1.3 μM
Solubility
Solubility (25C)* In vitro DMSO 9 mg/mL (25.98 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Return Policy Contact information
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High Purity Kinase Inhibitors on Signaling Pathways

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