ADL5859 HClCatalog No. A11072

Quick Overview

ADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM.
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ADL5859 HCl

Product Information
Catalog Num A11072
M. Wt 429
Formula C24H28N2O3.HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 850173-95-4
Synonyms ADL-5859
Chemical Name N,N-Diethyl-4-(5-hydroxyspiro[2H-1-benzopyran-2,4'-piperidin]-4-yl)benzamide hydrochloride
SMILES Code CCN(CC)C(=O)C1=CC=C(C=C1)C2=CC3(CCNCC3)OC4=C2C(=CC=C4)O.Cl

Biological activity
Introduction
ADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM.
Targets
δ-opioid receptor μ-opioid receptor κ-opioid receptor
0.8 nM(Ki)32 nM(Ki)37 nM(Ki)
Solubility
Solubility (25C) * In vitro DMSO 86 mg/mL (200.48 mM)
Water 5 mg/mL (11.65 mM)
Ethanol 1 mg/mL (2.33 mM)
In vivo 0.5% hydroxyethyl cellulose/0.1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Return Policy Contact information
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High Purity Kinase Inhibitors on Signaling Pathways

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