C646Catalog No. A12815

Quick Overview

C646 is a selective p300/CREB-binding protein (CBP) inhibitor (Ki = 400 nM).
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C646

Product Information
Catalog Num A12815
M. Wt 445.42
Formula C24H19N3O6
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 328968-36-1
Synonyms C 646, C-646
Chemical Name 4-[4-[[5-(4,5-Dimethyl-2-nitropheny?l)-2-furanyl]methylene]-4,5-dihydro-3-methyl-5-oxo?-1H-pyrazol-1-yl]benzoic acid
SMILES Code CC1=C(C=C(C(=C1)C2=CC=C(O2)/C=C\3/C(=NN(C3=O)C4=CC=C(C=C4)C(=O)O)C)[N+](=O)[O-])C

Biological activity
Introduction
C646 is a selective p300/CREB-binding protein (CBP) inhibitor (Ki = 400 nM).
Targets
p300/CBP (Cell-free assay)
400 nM(Ki)
Solubility
Solubility (25C) * In vitro DMSO 13 mg/mL (29.18 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Return Policy Contact information
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High Purity Kinase Inhibitors on Signaling Pathways

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