Ligand-gated Ion Channels

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Catalog No. Product Name Application Product Information
A10006 SALE

(-)-Huperzine A

GluR inhibitor
(-)-Huperzine A is a naturally occurring sesquiterpene alkaloid compound found in the firmoss Huperzia serrata.


GABAA agonist
Bretazenil, a benzodiazepine receptor partial agonist, as an adjunct in the prophylactic treatment of OP poisoning.


Felbamate is an antagonist at the NMDA-associated glycine binding site.

Gabapentin Hydrochloride

Gabapentin Hydrochloride is a GABA analogue.

GW791343 HCl

P2X7 modulator
GW791343 HCl acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2) and a positive allosteric modulator of rat P2X7.
A10490 SALE


Ivermectin is a broad-spectrum antiparasitic avermectin medicine.
A11873 SALE


Lamotrigine is a phenyltriazine sodium channel protein inhibitor of presynaptic neurons.
A11708 SALE

Memantine hydrochloride

Memantine hydrochloride is an antagonist at the NMDA receptor, binding to the ion channel site. it was used in the treatment of Parkinsonism.

Methyllycaconitine citrate

Methyllycaconitine citrate is a potent antagonist for ??7-containing neuronal nicotinic receptors (Ki = 1.4 nM). Interacts with ??4??2 and ??6??2 receptors at concentrations > 40 nM.

Ondansetron (Zofran)

Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic (to treat nausea and vomiting). Ondansetron reduces the activity of the vagus nerve, which deactivates the vomiting center in the medulla oblongata, and also blocks serotonin receptors in the chemoreceptor trigger zone.

Prasugrel (Effient)

Prasugrel is a novel platelet inhibitor used for the reduction of thrombotic cardiovascular events (including stent thrombosis) in patients with acute coronary syndrome who are to be managed with PCI.
A10966 SALE


Varenicline is a nicotinic receptor partial agonist.

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