Ligand-gated Ion Channels



12 Item(s)

per page

Set Descending Direction
Catalog No. Product Name Application Product Information
A10006

(-)-Huperzine A

GluR inhibitor
(-)-Huperzine A is a naturally occurring sesquiterpene alkaloid compound found in the firmoss Huperzia serrata.
A13784

Bretazenil

GABAA agonist
Bretazenil, a benzodiazepine receptor partial agonist, as an adjunct in the prophylactic treatment of OP poisoning.
A11862

Felbamate

-
Felbamate is an antagonist at the NMDA-associated glycine binding site.
A10414

Gabapentin Hydrochloride

-
Gabapentin Hydrochloride is a GABA analogue.
A11107

GW791343 HCl

P2X7 modulator
GW791343 HCl acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2) and a positive allosteric modulator of rat P2X7.
A10490

Ivermectin

-
Ivermectin is a broad-spectrum antiparasitic avermectin medicine.
A11873

Lamotrigine

-
Lamotrigine is a phenyltriazine sodium channel protein inhibitor of presynaptic neurons.
A11708

Memantine hydrochloride

-
Memantine hydrochloride is an antagonist at the NMDA receptor, binding to the ion channel site. it was used in the treatment of Parkinsonism.
A12681

Methyllycaconitine citrate

-
Methyllycaconitine citrate is a potent antagonist for ??7-containing neuronal nicotinic receptors (Ki = 1.4 nM). Interacts with ??4??2 and ??6??2 receptors at concentrations > 40 nM.
A11701

Ondansetron (Zofran)

-
Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic (to treat nausea and vomiting). Ondansetron reduces the activity of the vagus nerve, which deactivates the vomiting center in the medulla oblongata, and also blocks serotonin receptors in the chemoreceptor trigger zone.
A10748

Prasugrel (Effient)

-
Prasugrel is a novel platelet inhibitor used for the reduction of thrombotic cardiovascular events (including stent thrombosis) in patients with acute coronary syndrome who are to be managed with PCI.
A10966

Varenicline

-
Varenicline is a nicotinic receptor partial agonist.

12 Item(s)

per page

Set Descending Direction