Neurokinin Receptors



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Catalog No. Product Name Application Product Information
A11069

Fosaprepitant dimeglumine

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Fosaprepitant is a selective neurokinin-1 (NK-1) receptor antahonist.
A13103

GW679769 (Casopitant)

NK1 receptor antagonist
Casopitant mesylate is the mesylate salt of a centrally-acting neurokinin 1 (NK1) receptor antagonist with antidepressant and antiemetic activities.
A13104

Ibodutant (MEN 15596)

tachykinin NK2 receptor antagonist
Ibodutant is a tachykinin NK2 receptor antagonist for the treatment of Irritable Bowel Syndrome with diarrhoea (IBS-D)
A11756 SALE

MK-0517 (Fosaprepitant)

neurokinin-1 receptor antagonist
Fosaprepitant (MK-0517, L-758,298) is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.
A15187

NKP608

NK1 receptor antagonist
NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective, specific and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50=2.6 nM) and in vivo.
A15230 SALE

SB-222200

NK3 receptor antagonist
SB 222200 is a selective, reversible and competitive antagonist of human NK-3 receptor(Ki=4.4 nM) that effectively crosses the blood-brain barrier.
A15254

Talnetant

NK3 receptor antagonist
Talnetant is a potent and selective NK3 receptor antagonist(ki=1.4 nM, hNK-3-CHO); 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 uM.
A15255

Talnetant hydrochloride

NK3 receptor antagonist
Talnetant Hcl is a potent and selective NK3 receptor antagonist(ki=1.4 nM, hNK-3-CHO); 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 uM.
A12793

Vofopitant (GR 205171)

NK1 receptor antagonist
GR 205171 is a selective neurokinin-1 receptor antagonist

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