NMDA Receptors



11 Item(s)

per page

Set Descending Direction
Catalog No. Product Name Application Product Information
A12761

(+)-MK 801 Maleate

NMDA receptor antagonist
(+)-MK 801 is a potent antagonist of NMDA with Ki value of 30.5nM.
A13435

(-)-MK 801 maleate

NMDA receptor antagonist.
(-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel.
A15791

CGS19755

NMDA antagonist
CGS 19755 (cis-4-phosphonomethyl-2-piperidine carboxylic acid) was found to be a potent, stereospecific inhibitor of N-methyl-D-aspartate (NMDA)-evoked, but not KCl-evoked, [3H] acetylcholine release from slices of the rat striatum.
A12946

Eliprodil

NMDA antagonist
Eliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM).
A10251

Flupirtine maleate

NMDA antagonist
Non-opioid analgesic with muscle relaxant properties.
A15522

L-701324

NMDA/glycine receptor antagonist
L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor,
A13729

MDL 29951

NMDA receptor antagonist
MDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo.
A12751

NMDA

-
NMDA is a prototypic NMDA receptor agonist.
A12426

SDZ 220-581

NMDA receptor antagonist
SDZ 220-581 is a competitive NMDA receptor antagonist (pKi = 7.7).
A15235

SDZ 220-581 Ammonium salt

NMDA receptor antagonist
SDZ 220-581 ammonium salt is a potent, competitive antagonist at the NMDA glutamate receptor subtype(pKi= 7.7).
A11947

TCN 201

NMDA Receptor Antagonist
TCN 201 is a NMDA receptor antagonist selective for NR1/NR2A over NR1/NR2B-containing receptors

11 Item(s)

per page

Set Descending Direction