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Catalog No. Product Name Application Product Information
A13452

L161240

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L161240, was active against a P. aeruginosa construct in which the endogenous lpxC gene was inactivated and in which LpxC activity was supplied by the lpxC gene from E. coli.
A13472

Golotimod (SCV-07)

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Golotimod is an orally bioavailable synthetic peptide containing the amino acids D-glutamine and L-tryptophan connected by a gamma-glutamyl linkage with potential immunostimulating, antimicrobial and antineoplastic activities.
A13481

3,4-Dehydro Cilostazol

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3,4-Dehydro Cilostazol is a metabolite of Cilostazol.
A13482

4'-trans-Hydroxy Cilostazol

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4'-trans-Hydroxy Cilostazol is a metabolite of Cilostazol.
A13400

Bupranolol

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Bupranolol is a non-selective beta blocker without intrinsic sympathomimetic activity (ISA), but with strong membrane stabilizing activity.
A13416

Moxonidine Hydrochloride

imidazoline receptor 1 agonist
Moxonidine hydrochloride is a centrally acting antihypertensive agent.
A13418

Nisoxetine hydrochloride

Noradrenalin re-uptake inhibitor
Nisoxetine hydrochloride is a selective and potent inhibitor of norepinephrine transporter with little or no affinity for a range of other neurotransmitter receptors. Nisoxetine hydrochloride is an inhibitor of SLC6A2.
A14918

LH-RH, human

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LH-RH, human is a biochem/physiol Actions LHRH Hypothalamic peptide that stimulates release of gonadotrophins from anterior pituitary, thus regulating reproductive functions.
A14001

K-252a

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K-252a is a metabolite originally isolated from the culture broth of Nocardiopsis sp.. Experiments have shown that at high concentrations this compound is an ATP-competitive inhibitor of cyclic nucleotide-dependent protein kinases.
A13988

PR-104

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PR-104 is a non-toxic, small-molecule, hypoxia-activated, 3,5-dinitrobenzamide nitrogen mustard pre-prodrug with potential antitumor activity.
A13558

CHR-6494

Haspin inhibitor
CHR-6494 is a potent and selective Haspin (Haploid Germ Cell-Specific Nuclear Protein Kinase) inhibitor that blocks H3T3ph phosphorylation.
A13689 SALE

Exherin (ADH-1)

N-cadherin antagonist
Exherin is a small, cyclic pentapeptide vascular-targeting agent with potential antineoplastic and antiangiogenic activities.
A13701

NBMPR

ENT1 inhibitor
NBMPR is a nucleoside analog that competitively inhibits the equilibrative nucleoside transporter 1 (Kd = 0.1-1.0 nM, IC50s = 4.6 and 3.6 nM in rat and human, respectively).
A13649

Briciclib

cell cycle inhibitor
Briciclib is a benzyl styryl sulfone analog, and a disodium phosphate ester prodrug of ON 013100, with potential antineoplastic activity.
A13652 SALE

AVN-944

IMPDH inhibitor
AVN-944 is an orally available, synthetic small molecule with potential antineoplastic activity.
A13682 SALE

AHU-377 (Sacubitril calcium)

neprilysin inhibitor
AHU-377 is an inhibitor of neprilysin with IC50 value of 5nM.
A13610

5-Bromo Brassinin

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5-Bromo Brassinin is a derivative of Brassinin.
A13616

7-Methyluric Acid

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7-Methyluric Acid is a metabolite of Theobromine.
A13619

3-Methylcrotonyl Glycine

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3-Methylcrotonyl Glycine is a metabolite found in 3-methylcrotonylglycinuria, a metabolic disorder.
A13621

6-Maleimido-1-hexanol

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6-Maleimido-1-hexanol is a maleimide compound with a pendant hexanol moiety.
A13624

cis-Urocanic acid

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cis-Urocanic acid is a major ultraviolet-absorbing component of the stratum corneum.
A13631

MIF Antagonist

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MIF antagonist is an inhibitor of the dopachrome tautomerase activity of MIF in vitro (IC50 = 7 M) and in cells (IC50 = 25 M).
A13632

2-HG (sodium salt)

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a-Hydroxyglutaric acid (2-HG) is an a-hydroxy acid. It is normally metabolized to 2-oxoglutarate by D- and L-2-hydroxyglutarate dehydrogenases, and mutations in these enzymes cause 2-hydroxyglutaric aciduria, a neurometabolic disorder.
A13569

GZ-793A

VMAT2 inhibitor
GZ-793A is a selective inhibitor of vesicular monoamine transporter 2 (VMAT2), which transports the monoamine neurotransmitters from cellular cytosol into synaptic vesicles.
A13609

N-(p-Coumaroyl) Serotonin

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N-(p-Coumaroyl) Serotonin is an antibacterial agent which inhibits the production of proinflammatory cytokines by LPS-stimulated human blood monocytes.
A13535

R-121919

CRF1 receptor antagonist
R121919 is a potent small-molecule CRF1 receptor antagonist.
A13538

PKR Inhibitor

PKR Inhibitor
PKR Inhibitor is an oxindole/imidazole derivative that binds the ATP-binding site of PKR and blocks autophosphorylation with an IC50 value of 186-210 nM.3 PKR Inhibitor protects human neuroblastoma cells against cell damage triggered by tunicamycin-mediated endoplasmic reticulum stress.
A13541

EC-17

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EC-17 is a conjugate consisting of fluorescein isothiocyanate (FITC) conjugated with folate with potential antineoplastic activity.
A14924

Anisole Methoxybenzene

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Anisole methoxybenzene is a colorless liquid with a smell reminiscent of anise seed, and in fact many of its derivatives are found in natural and artificial fragrances.
A14131

NB-598

squalene epoxidase inhibitor
NB-598 is a potent competitive inhibitor of squalene epoxidase.
A13122

Amsilarotene (TAC-101)

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Amsilarotene (TAC-101) is a retinobenzoic acid with potential antineoplastic activity.
A13032 SALE

AT 56

L-PGDS inhibitor
AT-56 is am orally active inhibitor of lipocalin-type prostaglandin D synthase (L-PGDS) (Ki = 75 μM, IC50 = 95 μM).
A13230

TP808

-
N/A
A13455

GSK369796

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Shows antimalerial activity with IC50 values of 11.2 nM for 3D7 strain, 12.6 nM for HB3 strain, 17.6 nM for K1 strain
A13516

Coluracetam

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Coluracetam(MKC-231) is a new choline uptake enhancer.
A13520

Isatoribine monohydrate

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Isatoribine monohydrate is a novel guanosine analogue showing immunostimulatory activity both in vivo and in vitro. This compound acts on different components of the immune system including B cells, natural killer (NK) cells and antigen-presenting cells (APC).
A13642

Etofenamate

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Etofenamate is an anti-inflammatory, anti-arrhythmic amino acid.
A13663

Nifuratel

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Nifuratel is used as an antibacterial, antifungal, and antiprotozoal (Trichomonas).
A13692

PTZ-343

-
PTZ-343 is a phenothiazine derivative with chemical name: sodium 3-(10H-phenothiazin-10-yl)propane-1-sulfonate.
A13732

TGR5-Receptor-Agonist

TGR5(GPCR19) agonist
TGR5 Receptor Agonist is a potent TGR5(GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).
A13733 SALE

NSI-189

-
NSI-189 is a nootropic and neurogenic research chemical derived from nicotinamide and pyrazine.
A13734

ZLN005

PGC-1α regulator
ZLN005 is a PGC-1α Transcriptional Regulator, which shoed some beneficialfEffects on diabetic db/db mice.
A13739 SALE

SCH 54292

GDP exchange inhibitor
SCH 54292 is a novel GDP exchange inhibitor
A13768

AdipoRon

AdipoR1 and AdipoR2 agonist
AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)
A13783

Tirofiban Hydrochloride Hydrate

GPIIb/IIIa antagonist
Tirofiban, Hydrochloride Hydrate is a specific nonpeptide platelet fibrinogen receptor (GPIIb/IIIa) antagonist.
A13764

ST 101(ZSET1446)

-
ST 101 (ZSET1446) is a novel cognitive enhancer that promotes hippocampal neurogenesis and ameliorates depressive behavior in olfactory bulbectomized mice.
A13807 SALE

BMS303141

ATP-citrate lyase inhibitor
BMS303141 is a potent inhibitor of ATP citrate lyase (ACL). BMS303141 inhibits lipid synthesis in HepG2 cells with an IC50 of 8 μM, and lowers plasma triglycerides in a murine hyperlipdemia model.
A13826 SALE

PTC-209

BMI-1 inhibitor
PTC-209 is a novel potent and selective BMI-1 inhibitor, targeting the BMI-1 self-renewal machinery with an IC50 of ~0.5 ?M.
A13324 SALE

BAY57-1293

helicase primase inhibitor
BAY 57-1293 is a potent helicase primase inhibitor. BAY 57-1293 inhibits replication of herpes simplex virus (HSV) type 1 and type 2 in the nanomolar range in vitro by abrogating the enzymatic activity of the viral primase-helicase complex.
A13331

laxogenin

-
N/A

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