Other inhibitors



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Catalog No. Product Name Application Product Information
A13124

SNT-207707

MC4-Receptor Antagonist
SNT-207707 is an oral MC4-Receptor Antagonist
A13235

NVP-231

CerK inhibitor
NVP-231 is a potent, specific, and reversible CerK inhibitor that competitively inhibits binding of ceramide to CerK.
A12895 SALE

Thiamet G

O-GlcNAcase inhibitor
Thiamet G is a potent, selective O-GlcNAcase inhibitor with Kiof 21 nM, while exhibiting 37,000-fold selectivity over human lysosomal-hexosaminidase.
A13242

Quinacrine 2HCl

-
Quinacrine 2HCl is a histamine N-methyltransferase inhibitor
A13243 SALE

Apramycin Sulfate

protein synthesis inhibitor
Apramycin Sulfate is a broad spectrum aminocyclitol antibiotic and component of the Nebramycin complex, produced by a strain of Streptomyces tenebrarius
A13248 SALE

MGL-3196

thyroid hormone receptor agonist
MGL-3196 is an orally small-molecule liver-directed thyroid hormone receptor agonist designed to increase cholesterol uptake into the liver and increase its metabolism.
A13271

Fidaxomicin

-
Fidaxomicin is the major analogue of a family of macrocyclic lactones isolated independently by three different groups from cultures belonging to three different genera (Actinoplanes, Dactylosporangium and Micromonospora) known as lipiarmycin A3, tiacumicin B and clostomicin B1, respectively. Fidaxomicin is a narrow spectrum antibiotic with excellent activity against Gram positive bacteria, notably Clostridium difficile. Fidaxomicin acts in the gastrointestinal tract without undue disruption to gut microbial flora.
A13281

Pyrroloquinoline quinone

-
Pyrroloquinoline quinone is a cofactor of microbial quinoprotein enzyme, and imidazopyrroline. A redox/cofactor found in a a class of enzymes called quinoproteins.
A13297

Deferitrin (GT-56-252)

-
Deferitrin (GT-56-252) is the first drug in a class of desferrithiocin-derived hexadentate iron chelators.
A10016 SALE

5-Aminolevulinic acid hydrochloride

-
5-Aminolevulinic acid hydrochloride is a naturally occurring amino acid; precursor of tetrapyrroles in the biosynthesis of chlorophyll and heme.
A10581

Methyl Hesperidin

-
Methyl Hesperidin is a compound of the vitamin P group
A13354

Harmane

-
A13369 SALE

5-BrdU

-
5-BrdU is a synthetic thymidine analog; incorporated into DNA during replication. Used in assays for cell proliferation.
A13370

BCH

LAT1 inhibitor
BCH is an inhibitor of L-type amino acid transporter LAT1. Suppresses growth and induces apoptosis via activation of caspases in KB, Saos2 and C6 cancer cell lines.
A13404

FABP4 Inhibitor

-
FABP4 Inhibitor is a cell-permeable biphenylazolo-oxyacetate that acts as a potent and selective inhibitor of adipocyte Fatty-Acid-Binding Protein (aFABP/aP2) by targeting its fatty acid-binding pocket (Ki = < 2 nM in a competitive binding assay using 1,8-ANS), while exhibiting much lower affinity for muscle and epidermal FABP's (Ki = 250 nM and 350 nM, respectively).
A12908 SALE

Bioymifi

DR5 activator
Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.
A12910

Lupulone

-
Lupulone, a hop bitter acid, activates different death pathways involving apoptotic TRAIL-receptors, in human colon tumor cells and in their derived metastatic cells.
A13835 SALE

PF-06687859

DCPS inhibitor
RG3039 (PF-06687859) is orally bioavailable, brain-penetrant small molecule that has been shown to be an inhibitor of the mRNA decapping enzyme, DcpS.
A13887 SALE

TP-434 (Eravacycline)

-
TP-434 is a novel, broad-spectrum fluorocycline antibiotic with activity against bacteria expressing major antibiotic resistance mechanisms including tetracycline-specific efflux and ribosomal-protection.
A13966

TPT-260 (Dihydrochloride)

-
TPT-260 is a thiophene thiourea derivative.
A14052

YH249

-
N/A
A13134 SALE

CP-640186

acetyl-CoA carboxylase inhibitor
CP-640186 is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor with IC50s of 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively; with improved metabolic stability vs CP-610431.
A13746

FAI (5S rRNA modificator)

rRNA modificator
N/A
A13046 SALE

N6022

GSNOR inhibitor
N6022 is a potent, specific, and fully reversible inhibitor of S-nitrosoglutathione reductase (GSNOR) with an IC50 of 8 nM and a Ki of 2.5 nM.
A14157 SALE

AZD 7545

PDHK inhibitor
AZD7545 is a novel, selective small-molecule inhibitor of PDHK2 (PDH kinase2) with an IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2 respectively.
A14153

FH1 (BRD-K4477)

-
Enhances differentiation of induced pluripotent stem cells (iPSCs) to hepatocytes; also promotes the maturation of iPSC-derived hepatocytes.
A14144

FYX 051

XOR Inhibitor
Topiroxostat(FYX-051) is a novel and potent xanthine oxidoreductase (XOR) inhibitor with IC50 value of 5.3 nM.
A14061

Tomeglovir

-
Tomeglovir is a novel nonnucleosidic inhibitor of human cytomegalovirus replication.
A14074

Thymalfasin

-
N/A
A14077

Thymosin b4

-
Thymosin ??4 is naturally occuring, potent regulator of actin polymerization present in human platelets at a concentration of 200 - 500 uM.
A14123

FPH2 (BRD-9424)

-
FPH2 (BRD-9424) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.
A14140

TH 237A

neuroprotective agent
TH-237A is a novel neuroprotective agent, which possess protective properties against β-amyloid (Aβ)-induced neurodegeneration associated with Alzheimer's disease.
A11767

Bipenquinate

-
N/A
A13666 SALE

Gefarnate

-
Gefarnate is a synthetic isoprenoid that is used to treat chronic gastric and duodenic ulcers.
A14190 SALE

Tiplaxtinin (PAI-039)

PAI-1 inhbitor
Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.
A14098

Cyclazodone

-
Cyclazodone is a central stimulant with a mechanism of action similar to that of d-Amphetamine.
A14108

Picoplatin

-
Picoplatin is a new generation organic platinum analog with an extended spectrum of antineoplastic activity.
A14050

WW298

-
0
A14041

BMPS

-
BMPS is a short, sulfhydryl and amino reactive heterobifunctional crosslinking reagent.
A13990 SALE

Fosfluconazole

-
Fosfluconazole is a water-soluble phosphate prodrug of fluconazole - a triazole antifungal drug used in the treatment and prevention of superficial and systemic fungal infections.
A10861 SALE

Spectinomycin HCl

-
Spectinomycin is an antibiotic useful for the treatment of the bacterial infection, gonorrhea.
A13830 SALE

(S)-Reticuline

-
(S)-Reticuline is the (S)-enantiomer of Reticuline. An enantiomer of a tetrahydrobenzylisoquinoline alkaloid. Reticuline is a chemical compound found in a variety of plants including Lindera aggregata, Annona squamosa, and Ocotea fasciculata.
A13668

Levomefolate Calcium

-
Levomefolic acid is the primary biologically active form of folic acid used at the cellular level for DNA reproduction, the cysteine cycle and the regulation of homocysteine.
A13296

SP-420

-
SP-420 is an orally active small molecule that selectively binds iron and removes it from the body. In animal studies, SP-420 has shown excellent tissue penetration, highly efficient iron binding and a promising safety profile.
A13215 SALE

(Glp1)-Apelin-13

Apelin Receptor activator
(Glp1)-Apelin-13 is an activator of Apelin Receptor
A11821 SALE

Bindarit

MCP inhibitor
Bindarit is an anti-inflammatory small molecule that modulates the NFκB pathway.
A12002 SALE

Arctigenin

-
Arctigenin is an antioxidant, anti-inflammatory, antiproliferative and antiviral agent. It inhibits LPS-induced iNOS expression via inhibition of IκBα phosphorylation and p65 nuclear translocation (IC50 = 10 nM)
A11840 SALE

ENOblock (AP-III-a4)

-
ENOblock (AP-III-a4) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.
A12159

Ezatiostat

GSTP1-1 inhibitor
Ezatiostat is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity.
A12568

Tirasemtiv (CK-2017357)

fast-skeletal-troponin activator
Tirasemtiv amplifies skeletal muscle response to nerve activation in humans.

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