Other inhibitors



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Catalog No. Product Name Application Product Information
A13693

Gemcitabine elaidate

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Gemcitabine elaidate is a lipophilic, unsaturated fatty acid ester derivative of gemcitabine (dFdC), an antimetabolite deoxynucleoside analogue, with potential antineoplastic activity.
A13708 SALE

Atovaquone

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Atovaquone is an anti-protozoal mitochondrial electron transport inhibitor.
A13719 SALE

Treprostinil

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Treprostinil is a stable analog of prostacyclin that is used clinically for the treatment of PPH.
A14018

Chlorin E6

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Chlorin E6 is a natural molecule and a promising photosensitizer.
A13756

Cambendazole

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Cambendazole acts as an anthelmintic used in the treatment of Chagas’ disease.
A13279

Flurazepam dihydrochloride

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Flurazepam possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties.
A13300

Palosuran

Urotensin-II receptor antagonist
Palosuran is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.
A14111 SALE

Tafamidis (Fx1006A)

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Tafamidis is a potent and selective transthyretin kinetic stabilizer that inhibits the amyloid cascade.
A14926

DBU

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DBU is a chemical compound and belongs to the class of amidine compounds.
A15973

Lesinurad sodium

SUR/URAT1 inhibitor
Lesinurad is a selective uric acid re-absorption inhibitor (SURI) and is also a selective inhibitor of URAT1, a transporter in the kidney that regulates uric acid excretion from the body.
A15966

Hexaminolevulinate HCl

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Hexaminolevulinate HCl is the hexyl ester of 5-aminolevulinic acid (ALA) with photodynamic properties.
A13212

Eslicarbazepine Acetate

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Eslicarbazepine acetate is an antiepileptic drug.
A16082

BI 1467335 (PXS 4728A)

SSAO/VAP-1 inhibitor
PXS-4728A is a very potent and highly selective compound in development for the treatment of cardiometabolic diseases like the liver-related disease Nonalcoholic Steatohepatitis (NASH).
A16084

S3QEL 2

Complex III modulator
S3QEL 2 is a selective inhibitor of superoxide production from the outer Q-binding site of mitochondrial respiratory complex site III (IIIQo) without altering oxidative phosphorylation.
A16085

SPL-B

TACC3 inhibitor
SPL-B, Orally active inhibitor of transforming acidic coiled-coil protein (TACC3) that selectively inhibits the nucleation of centrosome microtubules in ovarian cancer cells, without affecting spindle assembly in normal cells.
A16093

BRD 7116

LSC inhibitor
BRD 7116 is a potent and selective Inhibitor of leukemia stem cell (LSC) activity (EC50 = 200 nM).
A16095

Propiolamide

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N/A
A16107

6-Carboxyfluorescein

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The single isomer, 6-Carboxyfluorescein, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid.
A16128

HA15

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HA15 is a molecule that targets specifically BiP/GRP78/HSPA5.
A16134

Hydroquinidine

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Hydroquinidine is an antiarrhythmic agent.
A16136

Molsidomine

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Molsidomine is an orally active, long acting vasodilating drug. Molsidomine is metabolized in the liver to the active metabolite linsidomine.
A16138

Sucralfate

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Sucralfate is a sucrose sulfate-aluminium complex that binds to the ulcer, creating a physical barrier that protects the gastrointestinal tract from stomach acid and prevents the degradation of mucus.
A16140

D panthenol

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D panthenol is an alcoholic analogue of D-pantothenic acid and cholinergic agent.
A16141

Oxybenzone

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Oxybenzone is an organic compound used in sunscreens; provides broad-spectrum ultraviolet coverage, including UVB and short-wave UVA rays.
A16145

Ciclesonide

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Ciclesonide is a glucocorticoid used to treat obstructive airway diseases.
A16148

Protirelin

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Protirelin is a thyrotropin-releasing hormone receptor used to treat hypothyroidism.
A16149

Ademetionine disulfate tosylate

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Ademetionine disulfate tosylate is a ubiquitous methyl donor involved in a wide variety of biological reactions, including those mediated by DNA and protein methyltransferases.
A15963

Fluoxymesterone

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Fluoxymesterone is an anabolic steroid with strong androgenic properties that has been used in the treatment of male hypogonadism, delayed puberty in males, and in the treatment of breast neoplasms in women.
A15962

Emeramide (BDTH2)

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Emeramide is a mercury and heavy metal chelator.
A16046

Hexa-D-arginine

furin inhibitor
Hexa-D-arginine is a inhibitor of furin (Ki values are 0.106, 0.58 and 13.2 uM for furin, PACE4 and PC1 respectively).
A15987

Sardomozide HCl

polyamine synthesis inhibitor
Sardomozide is a second-generation polyamine synthesis inhibitor, which inhibits the activity of the polyamine biosynthetic enzyme S-adenosylmethionine decarboxylase (SAMDC).
A15989

Sugammadex sodium

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Sugammadex soidum is an agent for reversal of neuromuscular blockade by the agent rocuronium in general anaesthesia.
A15994

WWL70

ABHD6 inhibitor
WWL70 is a potent inhibitor of α/β-hydrolase domain 6 (ABHD6) (IC50 = 70 nM), an enzyme which catalyzes the hydrolysis of 2-arachidonylglycerol.
A15995

Y-29794 Tosylate

PPCE inhibitor
Y-29794 Tosylate is an orally active, potent and specific non-peptide prolyl endopeptidase (PPCE) inhibitor.
A16006

4-Aminobenzoic acid

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4-Aminobenzoic acid is an intermediate in the synthesis of tetrahydrofolic acid in many non-mammalian organisms, including bacteria and fungi.
A16007

4-Aminoantipyrine

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4-Aminoantipyrine is a metabolite of aminopyrine with analgesic, anti-inflammatory, and antipyretic properties.
A16009

Iopamidol

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Iopamidol is a non-ionic, water-soluble radiographic contrast agent.
A16010

i-Inositol

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i-Inositol is a chemical compound which is sugar alcohol. i-Inositol is involved in a number of biological processes including insulin signal transduction, cytoskeleton transduction and so on.
A16013

Citric acid trilithium salt tetrahydrate

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Citric acid trilithium salt tetrahydrate is a pharmaceutical and construction material.
A10886

Cilastatin sodium

dipeptidase inhibitor
Cilastatin is a dipeptidase inhibitor that specifically inhibits DPEP1 (dehydrodipeptidase I), a renal membrane-bound glycoprotein involved in the hydrolytic metabolism of penem and carbapenem ??-lactam antibiotics.
A11282

PF-3644022

MK2 Inhibitor
PF-3644022 is a potent and selective mitogen-activated protein kinase (MAPK)-activated protein kinase-2 (MK2) inhibitor (Ki =3 nM).
A12788

Histone-H2A-(107-122)-Ac-OH

Histone-H2A peptide
Histone H2A is one of the five main histone proteins involved in the structure of chromatin in eukaryotic cells.
A16019

RETF-4NA

Selective chymase substrate
RETF-4NA is a chymase substrate peptide that is cleaved more avidly by α2-macroglobulin-bound chymase than the free, unbound form.
A16025

Y-29794 oxalate

Prolyl endopeptidase inhibitor
Y-29794 oxalate, inhibitor of prolyl endopeptidase, is a serine peptidase that may be implicated in the biosynthesis of amyloid β-peptide.
A16027

Decanoyl-RVKR-CMK

Proprotein convertases inhibitor
Decanoyl-RVKR-CMK is a selective, irreversible, and cell-permeable competitive inhibitor of proprotein convertases.
A16029

Butabindide oxalate

TPPII inhibitor
Butabindide oxalate is a selective and potent inhibitor of TPPII (tripeptidyl peptidase II).
A16033

CGS 35066

ECE inhibitor
CGS 35066 is a a potent endothelin-converting enzyme (ECE) inhibitor.
A16150 SALE

Azelaic acid

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Azelaic acid is an organic compound produced by the ozonolysis of oleic acid; component of a number of hair and skin conditioners.
A16151

Dehydrocholic acid

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Dehydrocholic acid is a synthetic bile acid, manufactured by the oxidation of cholic acid.
A16153

RS-1

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RS-1 is a RAD51-stimulatory compound, which increases the DNA binding activity of RAD51.

Items 151 to 200 of 635 total

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