Other inhibitors



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Catalog No. Product Name Application Product Information
A15631

Bucetin

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Bucetin is an analgesic and antipyretice agent with a risk of carcinogenesis.
A16090

Butamben

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Butamben is a long-duration local anesthetic used for the treatment of chronic pain.
A16383

2-Aminoheptane

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2-Aminoheptane is a nasal decongestant drug which is a sympathomimetic stimulant and vasoconstrictor.
A16384

4-Aminohippuric Acid

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4-Aminohippuric acid is a typical substrate of organic anion transport systems.
A16385

6-Acetamidohexanoic acid

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6-Acetamidohexanoic acid is a pharmaceutical intermediate.
A16388

Aceglutamide

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Aceglutamide is a psychostimulant, nootropic agent which functions as a prodrug to glutamine with improved potency and stability.
A16389

Acesulfame Potassium

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Acesulfame potassium is a non-nutritive sweetener.
A16391

Acetylleucine

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Acetylleucine is a drug used in the treatment of vertigo.
A16402

Aminoguanidine hydrochloride

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Aminoguanidine is a diamine oxidase and nitric oxide synthase inhibitor. It acts to reduce levels of advanced glycation end products (AGEs) through interacting with 3-deoxyglucosone.
A16412

Antimonyl potassium tartrate trihydrate

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Antimony potassium tartrate trihydrate is a powerful emetic, also used in the treatment of schistosomiasis and leishmaniasis.
A16415

Azaguanine-8

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Azaguanine-8 is a purine analogs showing antineoplastic activity by competing with guanine in the metabolism.
A16426

Carbazochrome sodium sulfonate(AC-17)

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Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for use in the treatment of hemorrhoids.
A16427

Carbimazole

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Carbimazole is an imidazole antithyroid agent.
A16430

Carzenide

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Carzenide is an organic synthesis intermediate, used for synthetic drug.
A16453

Cinchophen

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Cinchophen is an analgesic drug that is frequently used to treat gout.
A16456

Citiolone

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Citiolone is a derivative of the amino acid cysteine, used in liver therapy.
A16474

Cysteamine HCl

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Cysteamine is an agent for the treatment of nephropathic cystinosis and an antioxidant.
A14957

BRD7552

PDX1 inducer
BRD7552 is an inducer of transcription factor PDX1, which increases insulin expression.
A14939

Bisoctrizole

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Bisoctrizole is a broad-spectrum ultraviolet radiation absorber, absorbing UVB as well as UVA rays. Also a hybrid UV absorber, reflecting and scattering UV.
A14914

Bisacodyl

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Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement.
A16154

Sulisobenzone

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Sulisobenzone is an ingredient in some sunscreens which protects the skin from damage by UVB and short-wave UVA ultraviolet light.
A16158

Glutathione

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Glutathione acts as an antioxidant, a free radical scavenger and a detoxifying agent.
A16159

L-Tyrosine

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L-tyrosine is a non-essential amino acid. In animals it is synthesized from Ephenylalanine.
A16187

UR 1102

URAT1 inhibitor
UR 1102, inhibitor of the renal urate transporter URAT1 with high selectivity to URAT1 over OAT1 and OAT3 in vitro (Ki values 0.057 uM, 7.2 uM, and 2.4 uM, respectively), capable of increasing the fractional excretion of urinary uric acid, and reducing plasma uric acid more effectively than Benzbromarone.
A16191

ON-013100

cell cycle inhibitor
ON-013100 is a cell cycle inhibitor and is potentially useful for the treatment of mantle cell lymphoma.
A16200

Eprodisate Sodium

Fibrillogenesis inhibitor
Eprodisate is an orally available disodium salt form of eprodisate, a negatively charged sulfonated inhibitor of fibrillogenesis, that can be used in the treatment of amyloid A (AA) amyloidosis.
A16204

SCH00013

-
SCH00013 is a cardiotonic agent that primarily acts via an increase in myofibrillar Ca++ sensitivity, have a significant Ca(2+)sensitizing effect at pH 7.2 to 7.4.
A16205

WNK463

pan-WNK-kinase inhibitor
WNK463 is an orally bioavailable pan-WNK-kinase inhibitor.
A16206

Valbenazine

VMAT2 inhibitor
Valbenazine is a potent and selective VMAT2 inhibitor.
A16319

SecinH3

Cytohesin inhibitor
SecinH3 is a selective cytohesin inhibitor with IC50 of 2.4 μM, 5.4 μM, 5.4 μM, 5.6 μM, 5.6 μM, and 65 μM for hCyh2, hCyh1, mCyh3, hCyh3, drosophila steppke, and yGea2-S7, respectively.
A16321

3,3'-Diindolylmethane

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3,3'-Diindolylmethane(DIM) is a major digestive product of indole-3-carbinol, a potential anticancer component of cruciferous vegetables.
A16327

HMN-176

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HMN-176 is a stilbene derivative which inhibits mitosis without significant effect on tubulin polymerization.
A16331

AM-2394

glucokinase activator
AM-2394 is a structurally distinct glucokinase activator (GKA). AM-2394 activates glucokinase (GK) with an EC50 of 60 nM.
A16334

Necrosulfonamide

MLKL inhibitor
Necrosulfonamide is a pharmacological inhibitor of MLKL with IC50 values of 124 nM in human HT-29.
A16335

HTHQ

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HTHQ, which is a hydroquinone monoalkyl ether, is a potent anti-oxidative agent, even at low dose levels.
A14564

Benzyl alcohol

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Benzyl alcohol is an aromatic alcohol; a colorless liquid with a mild pleasant aromatic odor.
A14577

Benzyl benzoate

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Benzyl benzoate is one of the older preparations used to treat scabies. Scabies is a skin infection caused by the mite sarcoptes scabiei.
A16475

Cytidine

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Cytidine is a nucleoside molecule that is formed when cytosine is attached to a ribose ring, cytidine is a component of RNA.
A14931

Triisopropylsilane

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Triisopropylsilane is a highly selective reducing agent which can be used to prepare anti-1,2-diols.
A15242

sodium 4-pentynoate

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sodium 4-pentynoate is a alkynylacetate analogue; can be metabolically incorporated onto cellular proteins through biosynthetic mechanisms for profiling of acetylated proteins in diverse cell types.
A15244

Sodium formononetin-3'-sulfonate

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Sodium formononetin-3'-sulfonate is a water-sol. derivate of formononetin.
A15248

ST 2825

MyD88 dimerization Inhibitor
ST 2825 is a MyD88 pharmacologic inhibitor.
A15329

R18

14.3.3 proteins Antagonist
R18, antagonist of 14.3.3 proteins (KD ≈ 80 nM). Competitively inhibits 14.3.3-ligand interactions without requiring phosphorylation.
A15334

Plumbagin

Immunomodulators
Plumbagin, exhibits cytotoxicity in rodent models of carcinogenesis and carcinoma; has antifungal, antiviral, and antibacterial action.
A15339

iMAC2

Suppressor of mitochondrial apoptosis
iMAC2 inhibits mitochondrial apoptosis-induced channel (MAC) (IC50 = 28 nM).
A15425

Beta-Lipotropin (1-10), porcine

Morphine-like substance
Beta-lipotropin (beta-LPH) was found to contain within its C-terminal sequence the primary structure of these peptides.
A15521

AI-10-49

CBFBeta-SMMHC / RUNX1 inhibitor
AI-10-49 is a protein-protein interaction inhibitor that selectively binds to CBFβ-SMMHC and disrupts its binding to RUNX1 with a FRET IC50 of 0.26 uM,
A15539

NSC-41589

-
N/A
A15459

KRX-0402

DNA repair inhibitor
KRX-0402 is a small molecule that was specifically designed to block the DNA repair protein, MGMT. MGMT confers resistance to certain alkylating agents, such as temozolomide and BCNU, that are commonly used to treat brain cancer, melanoma and non-Hodgkin??s lymphoma.
A15464 SALE

SKQ1 Bromide

mitochondria-targeted antioxidant
SKQ1 is a potent mitochondria-targeted antioxidant. SKQ1 is also an API (active pharmaceutical ingredient) for making eye drop drug called Visomitin. SKQ1 showed activities (1) to prevent amyloid-beta-induced impairment of long-term potentiation in rat hippocampal slices.

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