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Peptide Receptors

Peptide Receptors

Catalog No.	Product Name	Application	Product Information
A12158	BIIE 0246	-	BIIE 0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM).
A13102	BMS-927711	CGRP receptor antagonist	BMS-927711 is a potent, selective, competitive human calcitonin gene-related peptide (CGRP) receptor antagonist that has shown in vivo efficacy without vasoconstrictor effect.
A12351	Desmopressin	-	Desmopressin is a synthetic vasopressin analog that acts as an agonist at V1B and V2 receptors (EC50 values are 11.4 and 23.9 nM and Ki values are 5.84 and 65.9 nM respectively).
A12646	Melanotan II	-	Melanotan II is a high affinity melanocortin receptor agonist (Ki values are 0.67, 6.6, 34 and 46 nM for MC1, MC4, MC3 and MC5 receptors respectively).
A10598	MK 3207 HCl	CGRP Receptor antagonist	MK 3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM. CGRP
A11255	MK-0974 (Telcagepant)	CGRP receptor antagonist	MK-0974 (Telcagepant) is a potent and selective antagonist of the human and rhesus CGRP receptors.
A12350	Ozarelix	GnRH antagonist	Ozarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors.
A12790	Parathyroid Hormone 1-34, Human	-	Human parathyroid hormone (hPTH) peptide fragment; contains the 34 N-terminal residues of hPTH. Agonist at parathyroid 1 (PTH1) and parathyroid 2 (PTH2) receptors.
A11820	Prostaglandin E1 (PGE1)	-	Prostaglandin E1 (PGE1) is the theoretical cyclooxygenase metabolite of dihomo-γ-linolenic acid (DGLA), but it is virtually undetectable in the plasma of normal humans or other animals. The IC50 of PGE1 for the inhibition of ADP-induced human platelet aggregation is 40 nM.
A11567	SB-408124	OX Receptor Antagonist	SB-408124 is a selective non-peptide orexin OX1 receptor antagonist (Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively). Blocks orexin-A induced grooming following oral administration in vivo. OX1 receptor
A12860	THIQ	-	THIQ is a potent and selective melanocortin 4 (MC4) receptor agonist (IC50 values are 1.2, 761 and 2067 nM for human MC4, MC3 and MC1 receptors respectively).
A11594	Tolvaptan	vasopressin receptor 2 antagonist	Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28?M. vasopressin receptor 2 vasopressin receptor 1a
A11979	YIL 781 Product Citations (1) D Lin ,etc. Abnormal response to the anorexic effect of GHS-R inhibitors and exenatide in male Snord116 deletion mouse model for Prader-Willi syndrome. Endocrinology, 2014, 155(7), 2355-2362.	-	YIL 781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM)