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Peptide Receptors

Peptide Receptors

Catalog No.	Product Name	Application	Product Information
A11979	YIL 781	-	YIL 781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) Product Citations (1) D Lin ,etc. Abnormal response to the anorexic effect of GHS-R inhibitors and exenatide in male Snord116 deletion mouse model for Prader-Willi syndrome. Endocrinology, 2014, 155(7), 2355-2362.
A12350	Ozarelix	GnRH antagonist	Ozarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors.
A12158	BIIE 0246	-	BIIE 0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM).
A12646	Melanotan II	-	Melanotan II is a high affinity melanocortin receptor agonist (Ki values are 0.67, 6.6, 34 and 46 nM for MC1, MC4, MC3 and MC5 receptors respectively).
A12790 SALE	Parathyroid Hormone 1-34, Human	-	Human parathyroid hormone (hPTH) peptide fragment; contains the 34 N-terminal residues of hPTH. Agonist at parathyroid 1 (PTH1) and parathyroid 2 (PTH2) receptors.
A12860	THIQ	-	THIQ is a potent and selective melanocortin 4 (MC4) receptor agonist (IC50 values are 1.2, 761 and 2067 nM for human MC4, MC3 and MC1 receptors respectively).
A11820 SALE	Prostaglandin E1 (PGE1)	-	Prostaglandin E1 (PGE1) is the theoretical cyclooxygenase metabolite of dihomo-γ-linolenic acid (DGLA), but it is virtually undetectable in the plasma of normal humans or other animals. The IC50 of PGE1 for the inhibition of ADP-induced human platelet aggregation is 40 nM.