All 'Androgen Receptor' Products



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Catalog No. Product Name Application Product Information
A10076

Andarine (GTX-007)

Androgen Receptor agonist
Andarine (GTX-007) is an investigational selective androgen receptor modulator (SARM).
A11923

ARN-509

Androgen Receptor inhibitor
ARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes.
A12396

AZD3514

AR inhibitor downregulator
AZD-3514 is a potent androgen receptor downregulator with potential anticancer cancer activity.
A10142

Bicalutamide (Casodex)

Androgen Receptor antagonist
Bicalutamide is an oral non-steroidal anti-androgen used in the treatment of prostate cancer and hirsutism.
A11409

Cyproterone acetate

Androgen Receptor antagonist
Cyproterone acetate is a synthetic derivative of 17-hydroxyprogesterone, and acts as an androgen receptor antagonist as well as a weak progesterone receptor agonist with weak progestational and glucocorticoid activity.
A10296

Dehydroepiandrosterone

-
Dehydroepiandrosterone is an important endogenous steroid hormone.
A15814

EPI-001

Androgen Receptor antagonist
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 ?M)
A10402

Flutamide

Androgen receptor antagonist
Flutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer.
A10562

MDV3100

Androgen receptor antagonist
MDV3100 is androgen-receptor inhibitor. Highly recommended inhibitor in AR research.
A10563

Megestrol Acetate

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Megestrol Acetate is a progesterone derivative with antineoplastic properties
A15797

ODM-201

Androgen receptor antagonist
ODM-201 is a potent and full antagonists for human AR (hAR) with IC50 values of 26 nM by transactivation assays in AR-HEK293 cells.
A11138

TOK-001 (Galeterone)

CYP17 inhibitor
TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor.

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