tankyrase (TNKS)

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  1. Inhibitor (5)


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Catalog No. Product Name Application Product Information
A15873

AZ6102

TNKS1/2 inhibitor
AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.
A15528

G007-LK

TNKS inhibitor
G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice,
A13731

JW 55

TNKS1/2 inhibitor
JW 55 is an inhibitor of the PARP domain of tankyrase 1 and 2 (TNKS1/2).
A15927

MN-64

TNKS inhibitor
MN-64 is a potent and selective inhibitor of Tankyrase 1 and 2 (IC50 = 6 and 72 nM, respectively).
A15786

NVP-TNKS656

TNKS2 inhibitor
NVP-TNKS656 is a highly potent, selective, and orally active TNKS2 inhibitor with IC50 of 6 nM; > 300 fold selectivity against PARP1 and PARP2.

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