TRPV



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Catalog No. Product Name Application Product Information
A13497

A-889425

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A-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human).
A12727 SALE

AMG517

TRPV1 antagonist
AMG 517 is a potent and selective TRPV1 antagonist.
A15496

Linoleylethanolamide

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Linoleylethanolamide is an endocannabinoid that also binds to TRPV1 (Ki = 5.60 ??M).
A15778

Mavatrep

TRPV1 antagonist
Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 ??M) of CYP isoforms 3A4, 1A2, and 2D6.
A15498

MRS1477

TRPV1 modulator
MRS1477 is a TRPV1 positive allosteric modulator.
A15830

RQ-00203078

TRPM8 antagonist
RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively), exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1.
A11143 SALE

SB-705498

TRPV1 antagonist
SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist.
A15857

SB366791

TRPV1 receptor antagonist
SB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist.

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