TRPV



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Catalog No. Product Name Application Product Information
A11143 SALE

SB-705498

TRPV1 antagonist
SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist.
A15857

SB366791

TRPV1 receptor antagonist
SB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist.
A15778

Mavatrep

TRPV1 antagonist
Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6.
A15498

MRS1477

TRPV1 modulator
MRS1477 is a TRPV1 positive allosteric modulator.
A15496

Linoleyl ethanolamide

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Linoleylethanolamide is an endocannabinoid that also binds to TRPV1 (Ki = 5.60 uM).
A13497

A-889425

TRPV1 receptor antagonist
A-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human).
A12727 SALE

AMG517

TRPV1 antagonist
AMG 517 is a potent and selective TRPV1 antagonist.
A14003

Resiniferatoxin

vanilloid receptor agonist
Resiniferatoxin is a natural analog of capsaicin (Item No. 92350) isolated from some plants of the genus Euphorbia, including E. resinifera.
A14201

GSK-2193874

TRPV4 blocker
GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
A15854

GSK1016790A

TRPV4 Activator
GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells.
A16423

(+)-Camphor

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Camphor is a waxy, flammable, white or transparent solid with a strong aroma, often used to relieve pain, reduce itching and treat fungal infections. It can activate TRPV1 and TRPV3

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