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$0.00 Biological Activity
Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors.
Targets
| Target | Value |
|---|---|
| 5-HT2C | pki: 10.46 |
| 5-HT2A | pki: 10.15 |
| 5-HT7 | pki: 9.94 |
| 5-HT2B | pki: 9.75 |
| 5-HT6 | pki: 9.6 |
| α2B-adrenergicreceptor | pki: 9.49 |
| D3receptor | pki: 9.38 |
| H1receptor | pki: 9 |
| D4receptor | pki: 8.95 |
| α1A-adrenergicreceptor | pki: 8.93 |
| α2C-adrenergicreceptor | pki: 8.91 |
| D2LReceptor | pki: 8.9 |
| α2A-adrenergicreceptor | pki: 8.9 |
| D1receptor | pki: 8.85 |
| 5-HT5A | pki: 8.84 |
| D2SReceptor | pki: 8.84 |
| 5-HT1A | pki: 8.6 |
| 5-HT1B | pki: 8.4 |
| H2receptor | pki: 8.21 |
| In vitro | DMSO | 78 mg/mL (194.1 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 24.89 mL | 124.43 mL | 248.86 mL |
| 0.5 mM | 4.98 mL | 24.89 mL | 49.77 mL |
| 1 mM | 2.49 mL | 12.44 mL | 24.89 mL |
| 5 mM | 0.5 mL | 2.49 mL | 4.98 mL |
*The above data is based on the productmolecular weight 401.84. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A10091 |
|---|---|
| Actions | Antagonist |
| CAS No. | 85650-56-2 |
| Formula | C17H16ClNO.C4H4O4 |
| M. Wt | 401.84 |
| Solubility | DMSO |
| Purity | >98% |
| SMILES | CN1C[[email protected]]2[[email protected]](C1)C3=C(C=CC(=C3)Cl)OC4=CC=CC=C24.C(=C\C(=O)O)\C(=O)O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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