Biological Activity
BIBX 1382 is a cell-permeable pyrimidopyrimidine compound that acts as a potent, reversible, ATP-competitive, and highly selective inhibitor of EGFR.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 21.7 mL | 108.51 mL | 217.01 mL |
0.5 mM | 4.34 mL | 21.7 mL | 43.4 mL |
1 mM | 2.17 mL | 10.85 mL | 21.7 mL |
5 mM | 0.43 mL | 2.17 mL | 4.34 mL |
*The above data is based on the productmolecular weight 460.8 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A11334 |
---|---|
Actions | Inhibitor |
CAS No. | 196612-93-8 |
Formula | C18H19ClFN7.2HCl |
M. Wt | 460.8 |
Purity | >98% |
Synonyms | BIBX1382, BIBX-1382 |
SMILES | CN1CCC(CC1)NC2=NC=C3C(=N2)C(=NC=N3)NC4=CC(=C(C=C4)F)Cl.Cl.Cl |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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