c-Ret

Catalog No.Inhibitor Name c-RETOther
A10250Regorafenib
****
Raf-1,VEGFR2,Kit
A10715Danusertib
**
Aurora A,Abl,TrkA
A11180TG101209
***
JAK2,FLT3,JAK3
A13832RPI-1
*

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. Regorafenib monohydrate

    Catalog No. A15218
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    Tyrosine kinase inhibitor
    Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively. Learn More

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