Canertinib (CI-1033)

Catalog No.: A10211
HER2/ErbB2 inhibitor
Canertinib (CI-1033) is an irreversible tyrosine-kinase inhibitor with activity against EGFR (IC50 0.8 nM), HER-2 (IC50 19 nM) and ErbB-4 (IC50 7 nM).
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Canertinib 10mg
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Canertinib 50mg
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Canertinib 200mg
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Adooq Products cited in reputable paper
Adooq's Canertinib (CI-1033) has been cited by 1 publications
  • Fukuda N, .et al. , ACS Synth Biol., 2015, 4(4):421-9 PMID: 25006755
  • Biological Activity
    Discription Canertinib (CI-1033) is an irreversible tyrosine-kinase inhibitor with activity against EGFR (IC50 0.8 nM), HER-2 (IC50 19 nM) and ErbB-4 (IC50 7 nM).
    Target Value
    Product Information
    Catalog Num A10211
    Formula C24H25ClFN5O3
    Molecular Weight 485.9
    CAS Number 267243-28-7
    Synonyms PD-183805

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    In vitro (25°C) DMSO 2 mg/mL (4.11 mM)
    Water Insoluble
    Ethanol 8 mg/mL (16.46 mM)
    In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 9 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 20.58 mL 102.9 mL 205.8 mL
    0.5 mM 4.12 mL 20.58 mL 41.16 mL
    1 mM 2.06 mL 10.29 mL 20.58 mL
    5 mM 0.41 mL 2.06 mL 4.12 mL
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    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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