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$0.00 Search results for 'am 2201'
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Verapamil
Catalog No. A12679 Verapamil is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor. Learn More -
Sulfamethoxazole sodium
Catalog No. A17452 Sulfamethoxazole sodium is an antibiotic used for bacterial infections. Learn More -
Ranitidine
Catalog No. A17721 Ranitidine is a potent, selective and orally active histamine H2-receptor antagonist with an IC50 of 3.3 μM that inhibits gastric secretion. Learn More -
Remimazolam
Catalog No. A22200 benzodiazepine derivative drugRemimazolam, also known as CNS-7056, is a benzodiazepine derivative drug, developed by PAION, in collaboration with Japanese licensee Ono Pharmaceutical as an alternative to the short-acting imidazobenzodiazepine midazolam, for use in induction of anaesthesia and conscious sedation for minor invasive procedures. Learn More -
Pemafibrate
Catalog No. A22201 PPAR alpha agonistPemafibrate, also known as (R)-K 13675, is a PPAR alpha agonist. Learn More -
Durlobactam sodium
Catalog No. A13801 beta-lactamase inhibitor drug candidateDurlobactam, also known as ETX2514, is a beta-lactamase inhibitor drug candidate. Learn More -
Ozogamicin
Catalog No. A12672 antibody-drug conjugate LinkerOzogamicin is an antibody-drug conjugate Linker. Learn More -
Dehydroascorbic acid
Catalog No. A12366 potent cerebroprotectionDehydroascorbic acid, a blood-brain barrier transportable form of vitamin C, mediates potent cerebroprotection in experimental stroke. Learn More -
Emedastine
Catalog No. A22158 histamine H1 receptor antagonistEmedastine is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM. Learn More -
Laninamivir octanoate
Catalog No. A22166 neuraminidase (NA) inhibitorLaninamivir octanoate (CS-8958), a prodrug of Laninamivir, is a long-acting neuraminidase (NA) inhibitor with anti-influenza virus activity. Learn More -
Lycorine
Catalog No. A22170 SCAP inhibitorLycorine is a natural alkaloid extracted from the Amaryllidaceae plant. Lycorine is a potent and orally active SCAP inhibitor with a Kd value 15.24 nM. Learn More -
Gentiopicroside
Catalog No. A22172 antianti-inflammatoryand antioxidative effectsGentiopicroside, a naturally occurring iridoid glycoside, inhibits P450 activity, with an IC50 and a Ki of 61 ?M and 22.8 ?M for CYP2A6; Gentiopicroside has antianti-inflammatoryand antioxidative effects. Learn More -
Eleutheroside B1
Catalog No. A22173 anti-human influenza virus efficacyEleutheroside B1, a coumarin compound, has a wide spectrum of anti-human influenza virus efficacy, with an IC50 value of 64-125 ?g/ml. Antiviral and anti-inflammatory activities. Learn More -
Oxyberberin
Catalog No. A22175 natural alkaloidBerlambine is a natural alkaloid isolated from many plants. Learn More -
BIO-013077-01
Catalog No. A22185 antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4BIO-013077-01, Novel potent antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4. Learn More -
Thiambutosine
Catalog No. A22187 candidate for treatment of lepromatous leprosyThiambutosine was a candidate for treatment of lepromatous leprosy. Learn More -
LY2828360
Catalog No. A22228 cannabinoid (CB2) agonistLY2828360 is a slowly acting but efficacious G protein-biased cannabinoid (CB2) agonist, inhibiting cAMP accumulation and activating ERK1/2 signaling. Learn More -
KN-93 phosphate
Catalog No. A22229 membrane-permeant synthetic inhibitorKN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM. Learn More -
Cl-amidine TFA
Catalog No. A22235 peptidylarginine deminase (PAD) inhibitorCl-amidine TFA is an orally active peptidylarginine deminase (PAD) inhibitor, with IC50 values of 0.8 μM, 6.2 μM and 5.9 μM for PAD1, PAD3, and PAD4, respectively. Learn More -
DS-1001b
Catalog No. A22236 mutant IDH-1 inhibitorDS-1001b is a mutant IDH-1 (Isocitrate Dehydrogenase-1) inhibitor extracted from patent WO2016052697A1, Example 168, and has antitumor activity. Learn More -
ML254
Catalog No. A22242 Positive Allosteric Modulators (PAMs)ML-254, also known as VU0430644; is Positive Allosteric Modulators (PAMs) of mGlu5 with Competitive MPEP-Site Interaction. Learn More -
CRT5
Catalog No. A22245 PKD inhibitorCRT5 (CRT0066051), a pyrazine benzamide, is a potent and selective PKD inhibitor with IC50 of 1 nM, 2 nM, and 1.5 nM for PKD1, PKD2, and PKD3, respectively. Learn More -
TAE-1
Catalog No. A22246 inhibitor of amyloid-β fibril formation and aggregationTAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. TAE-1 inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively. Learn More -
Enocyanin
Catalog No. A18660 anthocyanin extracted from grapesEnocyanin is an anthocyanin extracted from grapes. Enocyanin shows inhibitory effect on the leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase and esterase activity. Learn More -
Triphala
Catalog No. A16067 Anti-adipogenic, anti-inflammatory, and anti-neoplastic activitiesTriphala, an Ayurvedic polyherbal formulation comprising of equiproportional fruit parts of Terminalia chebula, Terminalia bellerica, and Phyllanthus emblica. Triphala inhibits NF-κB activation. Triphala exerts antifungal action. Anti-adipogenic, anti-inflammatory, and anti-neoplastic activities. Learn More -
Adenosine deaminase
Catalog No. A19330 Adenosine deaminase is an enzyme that catalyzes the irreversible deamination of adenosine and 2'-deoxyadenosine to inosine and 2'-deoxyinosine, respectively. Learn More -
Chitosan oligosaccharide
Catalog No. A20304 Chitosan oligosaccharide (COS) is an oligomer of β-(1??4)-linked D-glucosamine. Chitosan oligosaccharide (COS) activates AMPK and inhibits inflammatory signaling pathways including NF-κB and MAPK pathways. Learn More -
Hypotaurine
Catalog No. A20590 Hypotaurine (2-aminoethanesulfinic acid), an intermediate in taurine biosynthesis from cysteine in astrocytes, is an endogenous inhibitory amino acid of the glycine receptor. Learn More -
Hyaluronidase
Catalog No. A18232 local anesthetic additiveHyaluronidase (Hyaluronate 4-glycanohydrolase; Hyaluronoglucosaminidase) is a naturally occurring enzyme that depolymerizes hyaluronic acid by cleavage of glycosidic bonds and has been used as a local anesthetic additive. Learn More -
HM-43239
Catalog No. A20826 FLT3 inhibitorHM-43239 is a Novel Potent Small Molecule FLT3 Inhibitor, in Acute Myeloid Leukemia (AML) with FMS-like Tyrosine Kinase 3 (FLT3) Mutations Learn More -
Cinnamylamine
Catalog No. A20835 Cinnamylamine can be used for the preparation of Tranylcypromine, a drug that acts as a nonselective and irreversible inhibitor of the enzyme monoamine oxidase (MAO), and is used as an antidepressant and anxiolytic agent. Learn More -
Peptide 401
Catalog No. A13913 Peptide 401, a potent mast cell degranulating factor from bee venom, suppresses the increased vascular permeability due to intradermal injection of various smooth muscle spasmogens (histamine, and 5-HT). Learn More -
Exendin-4
Catalog No. A21580 glucagon-like peptide-1 receptor agonistExendin-4 (Exenatide), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. Learn More -
Apilimod mesylate
Catalog No. A22049 IL-12/IL-23 inhibitorApilimod (STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, and strongly inhibits IL-12 with IC50s of 1 nM and 2 nM, in IFN-γ/SAC-stimulated human PBMCs and SAC-treated monkey PBMCs, respectively. Learn More -
Sulopenem
Catalog No. A22051 beta-lactamase inhibitorSulopenem (CP-70429) is an orally active, potent inhibitor of beta-lactamase. Sulopenem is a parenteral penem antibiotic with broad-spectrum activities against Gram-positive and Gram-negative bacteria. Learn More -
TLR4-IN-C34
Catalog No. A22057 TLR4 inhibitorTLR4-IN-C34 is an orally active TLR4 inhibitor and reduces systemic inflammation in models of endotoxemia and necrotizing enterocolitis. Learn More -
H-β-Ala-AMC TFA
Catalog No. A22059 substrate for aminopeptidaseH-β-Ala-AMC TFA is a substrate for aminopeptidase. Learn More -
Filastatin
Catalog No. A22063 Candida albicans filamentation inhibitorFilastatin is a long-lasting inhibitor of Candida albicans filamentation. Filastatin inhibits adhesion by multiple pathogenic Candida species with an IC50 of ~3 μM in the GFP-based adhesion assay. Learn More -
Neuraminidase-IN-1
Catalog No. A22065 neuraminidase inhibitorNeuraminidase-IN-1 is a neuraminidase inhibitor, with an IC50 of 0.21 μM. Neuraminidase-IN-1 has excellent activity against H1N1 influenza virus. Learn More -
BAY 2416964
Catalog No. A22067 aryl hydrocarbon receptor (AHR) antagonistBAY 2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 192, has an IC50 of 341 nM. BAY 2416964 has the potential for solid tumors treatment. Learn More -
HS-243
Catalog No. A22071 transforming growth factor-?beta kinase inhibitorHS-243 is an inhibitor of transforming growth factor-?beta kinase. HS-243 can be used in treatment of cancer, malaria, inflammatory and other TAK1-?mediated diseases. Learn More -
PF9601N
Catalog No. A22075 monoamine oxidase B inhibitorPF9601N is a selective and potent monoamine oxidase B inhibitor that exhibit anti-Parkinsonian effects in several models of PD. Learn More -
BMS453
Catalog No. A22082 RARβ agonistBMS453 (BMS-189453), a synthetic retinoid, is a RARβ agonist and a RARα/RARγ antagonist. Learn More -
GW280264X
Catalog No. A22087 -
YM26734
Catalog No. A22091 rabbit platelet sPLA2 inhibitorYM-26734 is a rabbit platelet sPLA2 inhibitor that has been used to ameliorate local inflammatory responses in TPA-induced mouse ear edema. Learn More -
CYM 2503
Catalog No. A22092 positive allosteric modulator (PAM)CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. Learn More -
MCC950
Catalog No. A22097 inhibitor of NLRP3 (NOD-like receptor (NLR) familyMCC950 (CP-456773, CRID3) is a potent and selective inhibitor of NLRP3 (NOD-like receptor (NLR) family, pyrin domain-containing protein 3) with IC50 of 7.5 nM and 8.1 nM in BMDMs and HMDMs, respectively. Learn More -
BPU-11
Catalog No. A22101 HCN4 CLP ligandBPU-11 is a HCN4 CLP ligand. It acts by modulating channel function and completely abolishing the cAMP-induced shift in V1/2. Learn More
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