Search results for 'emd 1214063'

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  1. EMD-66684

    Catalog No. A22609
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    angiotensin II receptor antagonist
    EMD-66684 is a non-peptide angiotensin II receptor antagonist. Learn More
  2. Eniporide hydrochloride

    Catalog No. A21864
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    Na+/H+ exchange inhibitor
    Eniporide hydrochloride (EMD-96785 hydrochloride) is a potent Na+/H+ exchange inhibitor. Learn More
  3. Vilazodone Hydrochloride

    Catalog No. A11604
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    serotonin transporter (SER) inhibitor
    Vilazodone Hydrochloride (EMD 68843 Hydrochloride) is a serotonin transporter (SER) inhibitor and 5-HT1A receptor partial agonist. Learn More
  4. Rimeporide

    Catalog No. A17116
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    NHE-1 inhibitor
    Rimeporide (EMD-87580) is a potent and selective inhibitor of the Na+/H+ exchanger (NHE-1). Learn More
  5. Cilengitide trifluoroacetate

    Catalog No. A12371
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    Integrin inhibitor
    Cilengitide is a cyclic Arg-Gly-Asp peptide with potential antineoplastic activity. Cilengitide binds to and inhibits the activities of the alpha(v)beta(3) and alpha(v)beta(5) integrins, thereby inhibiting endothelial cell-cell interactions, endothelial cell-matrix interactions, and angiogenesis. Learn More
  6. Cilengitide

    Catalog No. A12372
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    Integrin inhibitor
    Cilengitide is a cyclic Arg-Gly-Asp peptide with potential antineoplastic activity. Cilengitide binds to and inhibits the activities of the alpha(v)beta(3) and alpha(v)beta(5) integrins, thereby inhibiting endothelial cell-cell interactions, endothelial cell-matrix interactions, and angiogenesis. Learn More
  7. Asimadoline

    Catalog No. A16920
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    KOR receptor
    Asimadoline is a potent κ-opioid receptor (KOR) agonist (IC50s = 5.6 and 1.2 nM for guinea pig and human receptors, respectively). Learn More
  8. Imeglimin hydrochloride

    Catalog No. A16283
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    oxidative phosphorylation blocker
    Imeglimin is the first in a new tetrahydrotriazine-containing class of oral antidiabetic agents, the glimins. It has been shown to act on the liver, muscle and pancreatic ??-cells to uniquely target the key defects of type 2 diabetes. Learn More
  9. Imeglimin

    Catalog No. A16282
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    oxidative phosphorylation blocker
    Imeglimin is an oxidative phosphorylation blocker that acts to inhibit hepatic gluconeogenesis, increase muscle glucose uptake, and restore normal insulin secretion. Learn More
  10. EMD534085

    Catalog No. A15956
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    Kinesin inhibitor
    EMD534085 is a kinesin inhibitor currently in clinical development. Learn More
  11. EMD638683

    Catalog No. A15079
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    SGK inhibitor
    EMD638683 is a potent inhibitor of SGK1 with an IC50 value of 3 uM. Learn More
  12. Safinamide

    Catalog No. A13294
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    MAO-B inhibitor
    Safinamide is a highly selective and reversible monoamine oxidase type B (MAO-B) inhibitor that increases neostriatal dopamine concentration. Learn More
  13. EMDT oxalate

    Catalog No. A19667
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    5-HT6 agonist
    EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects. Learn More
  14. Rislenemdaz

    Catalog No. A21907
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    NMDA receptor GluN2B antagonist
    Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. Learn More
  15. EMD638683 S-Form

    Catalog No. A11399
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    SGK1 inhibitor
    EMD638683 S-Form is the S-form of EMD638683. EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. Learn More
  16. EMD638683 R-Form

    Catalog No. A11398
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    SGK1 inhibitor
    EMD638683 R-Form is the R-form of EMD638683. EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. Learn More
  17. Remdesivir

    Catalog No. A17170
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    antiviral
    Remdesivir, also known as GS-5734, inhibits murine hepatitis virus (MHV) with an EC50 of 30 nM, and blocks SARS-CoV and MERS-CoV in HAE cells with EC50s of both 74 nM in HAE cells after treatment for 24 h. Learn More

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