Search results for 'glucagon receptor'

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  1. Glucagon-Like Peptide 1 (7-36) Amide

    Catalog No. A16895
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    Glucagon-Like Peptide 1 (7-36) Amide is a potent glucose-dependent insulinotropic peptide produced by post-translational processing of proglucagon in intestinal L-cells. Learn More
  2. Glucagon Human, His

    Catalog No. AP3258
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    Glucagon Human Recombinant, His Tag Learn More
  3. Glucagon Human

    Catalog No. AP3257
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    Glucagon Human Learn More
  4. Glucagon Human

    Catalog No. AP3256
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    Glucagon Human Recombinant Learn More
  5. Glucagon (19-29), human

    Catalog No. A14875
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    Ca 2+ /Mg 2+ -ATPase inhibitor
    Glucagon (19-29) (human) is a potent Ca 2+ /Mg 2+ -ATPase inhibitor. Learn More
  6. Sitagliptin phosphate monohydrate

    Catalog No. A10848
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    DDP-4 inhibitor
    Sitagliptin phosphate is an anti-diabetic (antihyperglycemic) drug of the dipeptidyl peptidase-4 (DPP-4) class. Inhibition of the enzyme DPP-4 is thought to increase Glucagon-like peptide-1 (GLP-1) which inhibits glucagon release , stimulates the insulin release and lowers blood glucose. Learn More
  7. Dulaglutide

    Catalog No. A16987
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    GLP-1 receptor agonist
    Dulaglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist. Learn More
  8. Liraglutide

    Catalog No. A16115
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    GLP-1 receptor agonist
    Liraglutide is a long-acting glucagon-like peptide-1(GLP-1) receptor agonist. Learn More
  9. BETP

    Catalog No. A13781
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    GLP-1 receptor agonist
    BETP is a selective positive allosteric modulator and partial agonist of the glucagon-like peptide 1 (GLP-1) receptor. Learn More
  10. GCGR Human

    Catalog No. AP3255
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    Glucagon Receptor Human Recombinant Learn More
  11. Lixisenatide

    Catalog No. A14076
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    GLP-1 receptor agonist
    ixisenatide inhibit glucagon release, markedly reduce postprandial glucago. have a promoting effct in diabetes mellitus (T2DM). Learn More
  12. MK 0893

    Catalog No. A11495
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    GCGR inhibitor
    MK 0893 is glucagon receptor antagonist as antidiabetic agents. Learn More
  13. Albiglutide

    Catalog No. A16823
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    GLP-1 agonist
    Albiglutide is a glucagon-like peptide-1 agonist (GLP-1 agonist). Learn More
  14. GLP 2 Human

    Catalog No. AP3254
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    Human Glucagon Like Peptide-2 Learn More
  15. GLP 1 Human

    Catalog No. AP3253
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    Human Glucagon Like Peptide-1 Learn More
  16. GLP-1 Human (31 a.a.)

    Catalog No. AP3252
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    Glucagon Like Peptide-1 (31 a.a.) Human Recombinant Learn More
  17. GLP 1 Human (37 a.a.)

    Catalog No. AP3251
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    Human Glucagon Like Peptide-1 (37 a.a.) Learn More
  18. Somatostatin

    Catalog No. A13453
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    Somatostatin is an endogenous peptide noted to inhibit the release of growth hormone, insulin and glucagon. Learn More
  19. AR-231453

    Catalog No. A13716
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    GPR119 agonist
    AR-231453 is a potent and selective small molecule agonis of GPR119 that enhances glucose dependent insulin secretion and glucagon like peptide-1 (GLP-1) release. Learn More
  20. Linagliptin (BI-1356)

    Catalog No. A11224
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    DPP-4 Inhibitor
    Linagliptin is a DPP-4 inhibitor, an enzyme that degrades the incretin hormones glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP). Learn More
  21. PF 06465469

    Catalog No. A17190
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    ITK inhibitor
    PF 06465469 is a potent the nonreceptor tyrosine kinase Itk (IL-2 inducible T-cell kinase) inhibitor. It also inhibits BTK. Learn More
    • New


    Catalog No. A17130
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    TNK2 inhibitor
    XMD16-5 is a tyrosine kinase nonreceptor 2(TNK2) inhibitor. Learn More
  22. S38093 HCl

    Catalog No. A17148
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    H3 receptors
    S38093 is an inverse agonist at histamine H3 receptors. CAS: 862896-30-8 (Free base) 1222097-72-4 (HCl) Learn More
  23. Cenicriviroc Mesylate

    Catalog No. A17028
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    CCR2/5 receptors inhibitor
    Cenicriviroc, also known as TAK-652 and TBR-652, is an inhibitor of CCR2 and CCR5 receptors, allowing it to function as an entry inhibitor which prevents the virus from entering into a human cell. CAS: 199673-74-0(LY 334370 hydrochloride); 182563-08-2 (LY 334370 Free Base) Learn More
  24. Lanifibranor

    Catalog No. A17041
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    PARP agonist
    Lanifibranor, also known as IVA-337, is a peroxisome proliferator-activated receptors (PPAR) agonist. Learn More
  25. WS 3

    Catalog No. A17047
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    TRPM8 agonist
    WS 3 is TRPM8 receptors agonist (EC50 = 3.7 μM) and cooling agent. Learn More
  26. RS 17053 HCl

    Catalog No. A16885
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    α1A antagonist
    RS 17053 HCl is α1A-adrenoceptor antagonist, with very high affinity for α1A receptors (pKi and pA2 estimates of 9.1 - 9.9) and a 30 - 100 fold selectivity over the α1B and α1D subtypes (pKi and pA2 estimates 7.7 - 7.8). Learn More
  27. SB399885 HCl

    Catalog No. A16971
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    SR-6 antagonist
    SB 399885 hydrochloride is a potent, brain penetrant, and orally active SR-6 antagonist. It displays > 200-fold selectivity for SR-6 over other serotonin receptors (pKi values are 9.11, 8.81 and 9.02 for human recombinant, native rat and native human SR-6 receptors, respectively). Learn More
  28. GSK4716

    Catalog No. A16956
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    ERRβ & ERRγ Agonist
    GSK4716 is an Estrogen-related receptors ERRβ and ERRγ agonist with minimal activity for ERRα, ERα and ERβ Learn More
  29. AZD-4635 (HTL1071)

    Catalog No. A16820
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    A2AR antagonist
    AZD-4635 (HTL1071) is an oral A2AR antagonist that binds to human A2AR with a Ki of 1.7 nM and with > 30-fold selectivity over other adenosine receptors. Learn More
  30. Proxyphylline

    Catalog No. A16821
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    A1 adenosine receptors antagonist
    Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets). Learn More
  31. TIGIT Human

    Catalog No. AP1720
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    T-Cell Immunoreceptor With Ig And ITIM Domains Human Recombinant Learn More
  32. Ro 25-6981 maleate

    Catalog No. A13144
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    NMDA receptors Blocker
    Ro 25-6981 is a high-affinity, potent and selective blocker of N-methyl- D-aspartate (NMDA) receptors. Learn More
  33. Vilanterol

    Catalog No. A13125
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    ultra-long-acting β₂ adrenoreceptor agonist
    Vilanterol is a novel and selective agonist of Beta2-AR with a PEC50 value of 10.37±0.05. Learn More
  34. Flunisolide

    Catalog No. A10398
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    Flunisolide is a corticosteroid often used to treat allergic rhinitis.The principal mechanism of action of Flunisolide is to activate glucocorticoid receptors, meaning it has an anti-inflammatory action. Learn More
  35. Acebutolol HCl

    Catalog No. A16387
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    β-adrenergic receptors antagonist
    Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias. Learn More
  36. Flavoxate

    Catalog No. A12900
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    Flavoxate binds and inhibits muscarinic receptors, thereby suppressing the micturition reflex and increases urinary bladder capacity by modifying the micturition center in the brain stem. Learn More
  37. VU 0364770

    Catalog No. A12139
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    mGlu4 receptors modulator
    VU 0364770 is a positive allosteric modulator at mGlu4 receptors with EC50 value of 290 nM in mGlu4-expressing HEK 293 cells. Learn More
  38. LOXO-101 sulfate

    Catalog No. A16239
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    TRK inhibitor
    LOXO-101 is a small molecule that was designed to block the ATP binding site of the TRK family of receptors, with 2 to 20 nM cellular potency against the TRKA, TRKB, and TRKC kinases. Learn More
  39. (S)-3,5-DHPG

    Catalog No. A16108
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    mGluR agonist
    (S)-3,5-DHPG is an agonist of the group I metabotropic glutamate receptors (mGluRs), binding both mGluR1a and mGluR5a (Ki = 0.9 and 3.9 uM, respectively) but not ionotropic glutamate receptors. Learn More
  40. Tretinoin

    Catalog No. A10944
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    RAR agonist
    Tretinoin is an endogenous agonist for retinoic acid receptors with IC50 value of 14 nM for RAR-alpha, RAR-beta and RAR-gamma receptors). Learn More
  41. BD-1047 2HBr

    Catalog No. A13196
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    Sigma-1 antagonist
    BD-1047 2HBr is a selective functional antagonist of sigma receptors, shows antipsychotic activity in animal models predictive of efficacy in schizophrenia. Learn More
  42. Ketanserin tartrate

    Catalog No. A13664
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    5HT2A antagonist
    Ketanserin tartrate is a salt of Ketanserin. Ketanserin is reported to have a high affinity for multiple G protein-coupled receptors, such as serotonin receptors. Learn More
  43. Cyclosporin H

    Catalog No. A15435
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    TPA/PMA inhibitor
    Cyclosporin H is a TPA/PMA inhibitor and a selective inhibitor of formyl peptide receptors (Ki = 0.1 uM). Learn More
  44. LY278584

    Catalog No. A15500
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    5-HT3 antagonist
    LY278584 is a potent and selective antagonist of 5-HT3 receptors. LY278584 is a useful ligand for studying the localization of 5-HT3 receptors in rat brain Learn More
  45. Imidafenacin

    Catalog No. A15490
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    M3 receptors inhibitor
    Imidafenacin is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). Learn More
  46. CIQ

    Catalog No. A15523
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    NMDA receptors Potentiator
    CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. Learn More
  47. N-Methylcytisine

    Catalog No. A15403
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    N-methylcytisine, a selective ligand of nicotinic receptors of acetylcholine in the CNS. Learn More
  48. Zolpidem

    Catalog No. A15288
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    Benzodiazepine agonist
    Zolpidem is an inhibitory neurotransmitter, by binding to GABAA receptors at the same location as benzodiazepines. Learn More
  49. SU14813 double bond Z

    Catalog No. A15250
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    VEGFR Inhibitor
    SU14813 is an oral, multitargeted tyrosine kinase inhibitor (TKI) targeting vascular endothelial growth factor receptors (VEGFR), platelet-derived growth factor receptors (PDGFR), Kit, and fms-like tyrosine kinase 3 (FLT-3). Learn More

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