Search results for 'jwh 307'

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  1. Higenamine

    Catalog No. A22315
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    β2-AR agonist
    Higenamine (Norcoclaurine), a β2-AR agonist, is a key component of the Chinese herb aconite root that prescribes for treating symptoms of heart failure in the oriental Asian countries. Learn More
  2. N6-Cyclopentyladenosine

    Catalog No. A19595
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    Adenosine A1 receptor agonist
    N6-Cyclopentyladenosine (CPA) is a selective Adenosine A1 receptor agonist, with Ki values of 2.3 nM, 790 nM and 43 nM for human A1, A2A and A3 receptors, respectively. Learn More
  3. Flumatinib

    Catalog No. A16258
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    multi-kinase inhibitor
    Flumatinib is a multi-kinase inhibitor with IC50 Values of 1.2 nM, 307.6 nM and 2662 nM for c-Abl, PDGFRbeta and c-Kit respectively. Learn More
  4. BIO-013077-01

    Catalog No. A22185
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    antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4
    BIO-013077-01, Novel potent antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4. Learn More
  5. (R)-Propranolol hydrochloride

    Catalog No. A22258
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    β-adrenergic receptor (βAR) antagonist
    (R)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol (HY-B0573). Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. Learn More
  6. RY785

    Catalog No. A22104
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    inhibitor of Kv2.1 and Kv2.2
    RY785 (Kv2-IN-A1) is an inhibitor of Kv2.1 and Kv2.2. Learn More
  7. LDN-193189 2HCl

    Catalog No. A22307
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    BMP signaling inhibitor
    LDN193189 HCl (DM-3189) is the hydrochloride salt of LDN193189, which is a selective BMP signaling inhibitor, and inhibits the transcriptional activity of the BMP type I receptors ALK2 and ALK3 with IC50 of 5 nM and 30 nM in C2C12 cell lines, respectively, 200-fold selectivity for BMP versus TGF-β. Learn More
  8. BTK inhibitor 1 (Compound 27)

    Catalog No. A22445
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    BTK inhibitor
    BTK inhibitor 1 (compound 27) is an inhibitor of BTK with an IC50 of 0.11 nM for Btk and inhibits B cell activation in hWB with an IC50 of 2 nM. Learn More
  9. GRA Ex-25

    Catalog No. A20625
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    glucagon receptor inhibitor
    GRA Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and human glucagon receptors, respectively. Learn More
  10. ST034307

    Catalog No. A20414
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    AC1 inhibitor
    ST034307 is a potent and selective adenylyl cyclase 1 (AC1) inhibitor, with IC50 of 2.3 μM. Learn More
  11. Simurosertib

    Catalog No. A20392
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    CDC7 inhibitor
    Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. Learn More
  12. Antifungal agent 1

    Catalog No. A20307
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    Antifungal agent 1 is a potent antifungal agent. Learn More
  13. Ds-HAPP

    Catalog No. A19307
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    Ds-HAPP is an anthrancenyl and dansyl fluorophore ligand. Learn More
  14. PLpro inhibitor

    Catalog No. A21044
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    Plpro inhibitor
    PLpro inhibitor is a potent inhibitor of papain-like protease (PLpro) with IC50 of 2.6 uM. Learn More
  15. (R)-Simurosertib

    Catalog No. A21894
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    CDC7 kinase inhibitor
    (R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. Learn More
  16. ATN-161

    Catalog No. A21307
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    integrin α5β1 antagonist
    ATN-161 is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. Learn More
  17. Emiglitate

    Catalog No. A20917
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    α-glucoside hydrolase inhibitor
    Emiglitate (BAY o 1248) is a potent, selective and competitive inhibitor of α-glucoside hydrolase. Learn More
  18. Diclofenac

    Catalog No. A17814
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    COX inhibitor
    Diclofenac is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor, with IC50s of 4 nM, 1.3 nM for human COX-1 and COX-2 in CHO cells, and 5.1, 0.84 μM for ovine COX-1 and COX-2, respectively. Learn More
  19. (4-Acetamidocyclohexyl) nitrate

    Catalog No. A13355
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    guanylate cyclase activator
    (4-Acetamidocyclohexyl) nitrate (BM121307) is a guanylate cyclase activator that was in phase I development for the treatment of ischaemic heart disorders. The research has been discontinued. Learn More
  20. Y-33075 dihydrochloride

    Catalog No. A11611
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    ROCK inhibitor
    Y-33075 dihydrochloride is a selective ROCK inhibitor with an IC50 of 3.6 nM. Learn More
  21. NMDI14

    Catalog No. A12958
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    NMD inhibitor
    NMDI14 is a nonsense mediated RNA decay (NMD) inhibitor. Learn More
  22. Ipenoxazone

    Catalog No. A12307
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    Ipenoxazone is a potent and centrally acting muscle relaxant. Learn More
  23. GSK2593074A

    Catalog No. A13600
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    necroptosis inhibitor
    GSK2593074A (GSK??074) is a necroptosis inhibitor with dual targeting ability to both RIP1 and RIP3. Learn More
  24. BAY885

    Catalog No. A13765
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    ERK5 inhibitor
    BAY885 is a novel ERK5 inhibitor. Learn More
  25. STF-083010

    Catalog No. A16720
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    IRE1α inhibitor
    STF-083010 is a specific IRE1α inhibitor. STF-083010 inhibits Ire1 endonuclease activity, without affecting its kinase activity, after endoplasmic reticulum stress. Learn More
  26. Levoleucovorin Calcium

    Catalog No. A11626
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    Levoleucovorin calcium is the calcium salt of Levoleucovorin, which is the enantiomerically active form of folinic acid. Learn More
  27. Enzaplatovir

    Catalog No. A20830
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    RSV fusion protein inhibitor
    Enzaplatovir is an inhibitor of Respiratory Syncytial Virus (RSV). It can be used as a viral fusion protein inhibitor. Learn More
  28. RTC-30

    Catalog No. A18865
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    RTC-30 is an optimized phenothiazine with anti-cancer potency. RTC-30 contains a hydroxylated linker (N) that confers increased oral bioavailability. Learn More
  29. NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). Learn More
  30. RTC-5

    Catalog No. A19067
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    RTC-5 is an optimized phenothiazine with anti-cancer potency. RTC-5 demonstrates efficacy against a xenograft model of an EGFR driven cancer, its effects is attributed to concomitant negative regulation of PI3K-AKT and RAS-ERK signaling. Learn More
  31. ODM-203

    Catalog No. A19098
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    FGFR/VEGFR inhibitor
    ODM-203 is a potent FGFR and VEGFR families inhibitor with IC50s of 11, 16, 6, 35 nM towards recombinant FGFR1, FGFR2, FGFR3 and FGFR4 as well as 26, 9, 5 nM towards VEGFR1, VEGFR2 and VEGFR3, respectively. Learn More
  32. LY-2940094

    Catalog No. A19125
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    NOP receptor antagonist
    LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. Learn More
  33. AN11251

    Catalog No. A19475
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    AN11251 is a potent and oral active anti-Wolbachia agent with potential for treatment of onchocerciasis and lymphatic filariasis, with EC50 values of 1.5 nM in LDW1 cell lines and 15 nM in C6/36 cell lines. Learn More
  34. ZXH-3-26

    Catalog No. A18399
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    PROTAC BRD4 degrader
    ZXH-3-26 is a selective PROTAC BRD4 degrader with a DC50/5h (DC50/5h referring to half-maximal degradation after 5 hours of treatment) of ~ 5 nM. Learn More
  35. GRL0617

    Catalog No. A18780
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    SARS PLPro inhibitor
    GRL0617 is a potent, selective and competitive noncovalent inhibitor of SARS PLPro, with an IC50 of 0.6 μM, and with a Ki of 0.49 μM. Learn More
  36. Metoclopramide hydrochloride hydrate

    Catalog No. A18072
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    Dopamine D2 antagonist
    Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. Learn More
  37. o-Cresol

    Catalog No. A17823
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    o-Cresol is a compound used as a disinfectant and have also been used as antiseptic in surgery. Learn More
  38. Revaprazan Hydrochloride

    Catalog No. A17506
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    Acid pump antagonist
    Revaprazan hydrochloride is a novel acid pump antagonist (APA). Revaprazan hydrochloride reduces COX-2 expression and has significant anti-inflammatory actions activities in H. pylori infection. Learn More
  39. Benznidazole

    Catalog No. A17307
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    Benznidazol (Ro 07-1051) is an antiparasitic medication, with an IC50 of 20.35 μM for Colombian T. cruzi strains, and has been used in the treatment of Chagas disease. Learn More
  40. Treponema TmpA 45kDa

    Catalog No. AP6307
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    Treponema pallidum TmpA, 45kDa Recombinant Learn More
  41. IL 16 Human, (121 a.a.)

    Catalog No. AP5307
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    Interleukin-16 Human Recombinant, (121 a.a.) Learn More
  42. GSTT1 Human

    Catalog No. AP4904
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    Glutathione S-Transferase Theta-1 Human Recombinant Learn More
  43. NAE1 Human

    Catalog No. AP4307
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    NEDD8 Activating Enzyme E1 Subunit 1 Human Recombinant Learn More
  44. Procalcitonin Mouse

    Catalog No. AP3307
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    Procalcitonin Mouse Recombinant Learn More
  45. CRABP2 Antibody

    Catalog No. AP3079
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    Cellular Retinoic Acid binding Protein 2, Mouse Anti Human Learn More
  46. FABP7 Antibody

    Catalog No. AP3078
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    Fatty Acid Binding Protein-7, Mouse Anti Human Learn More
  47. CFL1 Antibody

    Catalog No. AP3077
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    Cofilin-1, Mouse Anti Human Learn More
  48. BID Antibody

    Catalog No. AP3076
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    BH3 Interacting Domain Death Agonist , Mouse Anti Human Learn More
  49. VAMP3 Antibody

    Catalog No. AP3075
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    Synaptobrevin-3, Mouse Anti Human Learn More
  50. CHGA Antibody

    Catalog No. AP3074
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    Chromogranin-A, Mouse Anti Human Learn More

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