Biological Activity
CCT241533 is a potent and selective Inhibitor of CHK2 that potentiates the cytotoxicity of PARP inhibitors.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.61 mL | 113.07 mL | 226.14 mL |
0.5 mM | 4.52 mL | 22.61 mL | 45.23 mL |
1 mM | 2.26 mL | 11.31 mL | 22.61 mL |
5 mM | 0.45 mL | 2.26 mL | 4.52 mL |
*The above data is based on the productmolecular weight 442.2 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A11108 |
---|---|
Actions | Inhibitor |
CAS No. | 1262849-73-9 |
Formula | C23H27FN4O4 |
M. Wt | 442.2 |
Purity | >98% |
Synonyms | CCT-241533 |
SMILES | CC(C)([[email protected]@H]1CNC[[email protected]]1NC2=N/C(=C/3\C=C(C=CC3=O)F)/NC4=CC(=C(C=C42)OC)OC)O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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