Metabolism

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  1. MTP inhibitor

    PF-02575799 is a microsomal triglyceride transfer protein (MTP) inhibitor with an IC50 of 0.77±0.29 nM.

  2. MTP inhibitor

    Lomitapide is a potent microsomal triglyceride transfer protein (MTP) inhibitor.
  3. MTP inhibitor

    Implitapide (AEGR 427) is a microsomal triglyceride transfer protein (MTP) inhibitor.
  4. MTP inhibitor

    Lomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.

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