CFTR-Inhibitor-II

Catalog No.: A13723

CFTR inhibitor

CFTR-Inhibitor-II

CFTR-Inhibitor-II Chemical Structure

CAS NO. 328541-79-3

CFTR inhibitor II, also known as GlyH-101, is a glycine hydrazide that selectively and reversibly blocks the CFTR channel (Ki = 4.3 uM).

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25 mg
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Dao-Lai Zhang, .et al. Gq activity- and β-arrestin-1 scaffolding-mediated ADGRG2/CFTR coupling are required for male fertility, eLife, 2018, 7: e33432 PMID: 29393851

Biological Activity

CFTR inhibitor II, also known as GlyH-101, is a glycine hydrazide that selectively and reversibly blocks the CFTR channel (Ki = 4.3 uM).
Targets
CFTR
4.3 μM(Ki)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.28 mL 101.38 mL 202.76 mL
0.5 mM 4.06 mL 20.28 mL 40.55 mL
1 mM 2.03 mL 10.14 mL 20.28 mL
5 mM 0.41 mL 2.03 mL 4.06 mL

*The above data is based on the productmolecular weight 493.2. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13723
Actions Inhibitor
M. Wt 493.2
Formula C19H15Br2N3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 328541-79-3
Synonyms GlyH-101, Cystic Fibrosis Transmembrane Conductance, Regulator Inhibitor II
SMILES C1=CC=C2C=C(C=CC2=C1)NCC(=O)NN/C=C/3\C=C(C(=C(C3=O)Br)O)Br

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