CUDC-101

Catalog No.: A10246

HDAC inhibitor

CUDC-101

CUDC-101 Chemical Structure

CAS NO. 1012054-59-9

CUDC-101 is a novel compound which inhibits multiple targets, which is designed to inhibit HDAC, EGFR and Her2.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $70.00

Special Price $63.00

50 mg

Regular Price: $260.00

Special Price $234.00

100 mg

Regular Price: $480.00

Special Price $432.00

200 mg

Regular Price: $720.00

Special Price $648.00

10mM * 1mL in DMSO

Regular Price: $89.00

Special Price $80.10

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CUDC-101 is a novel compound which inhibits multiple targets, which is designed to inhibit HDAC, EGFR and Her2.
Targets
Target Value
EGFRIC50: 2.4nM
HDACIC50: 4.4nM
HDAC1IC50: 4.5nM
HDAC6IC50: 5.1nM
HDAC3IC50: 9.1nM
HDAC5IC50: 11.4nM
HDAC2IC50: 12.6nM
HDAC4IC50: 13.2nM
HER2IC50: 15.7nM
HDAC10IC50: 26.1nM
HDAC9IC50: 67.2nM
HDAC8IC50: 79.8nM
HDAC7IC50: 373nM
In vitro (25°C) DMSO 20 mg/mL (46.03 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.01 mL 115.07 mL 230.15 mL
0.5 mM 4.6 mL 23.01 mL 46.03 mL
1 mM 2.3 mL 11.51 mL 23.01 mL
5 mM 0.46 mL 2.3 mL 4.6 mL

*The above data is based on the productmolecular weight 434.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10246
Actions Inhibitor
M. Wt 434.5
Formula C24H26N4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1012054-59-9
Synonyms CUDC101
SMILES COC1=C(C=C2C(=C1)N=CN=C2NC3=CC=CC(=C3)C#C)OCCCCCCC(=O)NO

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy CUDC-101 | CUDC-101 Supplier | purchase CUDC-101 | CUDC-101 cost | CUDC-101 manufacturer | order CUDC-101 | CUDC-101 distributor | buy 1012054-59-9| 1012054-59-9 Supplier | purchase 1012054-59-9 | 1012054-59-9 cost | 1012054-59-9 manufacturer | order 1012054-59-9 | 1012054-59-9 distributor
Rewards