TG 100713

Catalog No. A11956

TG 100713 is an inhibitor of PI3-kinase that inhibits endothelial cell proliferation.
Catalog Num A11956
M. Wt 254.25
Formula C12H10N6O
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 925705-73-3
Synonyms TG100713
SMILES C1=CC(=CC(=C1)O)C2=CN=C3C(=N2)C(=NC(=N3)N)N
TG 100713 is an inhibitor of PI3-kinase that inhibits endothelial cell proliferation.
Targets
PI3Kδ PI3Kγ PI3Kα PI3Kβ
24 nM50 nM165 nM215 nM
In vitro DMSO 2 mg/mL (7.86 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 39.33 mL 196.66 mL 393.31 mL
0.5 mM 7.87 mL 39.33 mL 78.66 mL
1 mM 3.93 mL 19.67 mL 39.33 mL
5 mM 0.79 mL 3.93 mL 7.87 mL

*The above data is based on the productmolecular weight 254.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.