Elacestrant

Catalog No. A12244

Elacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.
Catalog Num A12244
M. Wt 458.63
Formula C30H38N2O2
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 722533-56-4
Synonyms RAD1901, RAD 1901, RAD-1901
SMILES OC1=CC=C2C[[email protected]](C3=CC=C(OC)C=C3N(CC)CC4=CC=C(CCNCC)C=C4)CCC2=C1
Elacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.8 mL 109.02 mL 218.04 mL
0.5 mM 4.36 mL 21.8 mL 43.61 mL
1 mM 2.18 mL 10.9 mL 21.8 mL
5 mM 0.44 mL 2.18 mL 4.36 mL

*The above data is based on the productmolecular weight 458.63. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.