A-1165442

Catalog No. A21516

A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1.
Catalog Num A21516
M. Wt 431.86
Formula C22H20ClF2N3O2
Purity >98%
Storage at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
CAS No. 1221443-94-2
Synonyms A1165442, A 1165442
SMILES O=C(NC1=CC=CC2=C1C=C(C)N=C2)N[[email protected]]3C4=CC=C(Cl)C=C4OC(CF)(CF)C3
A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.16 mL 115.78 mL 231.56 mL
0.5 mM 4.63 mL 23.16 mL 46.31 mL
1 mM 2.32 mL 11.58 mL 23.16 mL
5 mM 0.46 mL 2.32 mL 4.63 mL

*The above data is based on the productmolecular weight 431.86. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.