Crenigacestat (LY3039478)

Catalog No.: A13544
Notch inhibitor
LY3039478 is a orally bioavailable, novel small molecule Notch inhibitor with an IC50 of ~1nM in most of the tumor cell lines tested.
Grouped product items
Product Name Price Stock Qty
Crenigacestat (LY3039478) 5mg
$140.00
In stock
Crenigacestat (LY3039478) 10mg
$220.00
In stock
Crenigacestat (LY3039478) 25mg
$440.00
In stock
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Important Notice: For research use only. We do not sell to patients.

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Biological Activity
Discription LY3039478 is a orally bioavailable, novel small molecule Notch inhibitor with an IC50 of ~1nM in most of the tumor cell lines tested.
Product Information
Catalog Num A13544
Formula C22H23F3N4O4
Molecular Weight 464.43763
CAS Number 1421438-81-4
SMILES C[C@@H](C(=O)N[C@H]1C2=CC=CC=C2C3=C(N=CC=C3)N(C1=O)CCO)NC(=O)CCC(F)(F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 81 mg/mL (174.4 mM)
Water Insoluble
Ethanol 62 mg/mL (133.49 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.53 mL 107.66 mL 215.31 mL
0.5 mM 4.31 mL 21.53 mL 43.06 mL
1 mM 2.15 mL 10.77 mL 21.53 mL
5 mM 0.43 mL 2.15 mL 4.31 mL
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This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

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