PD168393
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | PD168393 is a potent, cell-permeable, irreversible inhibitor of EGFR with IC50 value of 700 pM. | ||
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Targets |
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Catalog Num | A12725 |
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Formula | C17H13BrN4O |
Molecular Weight | 369.22 |
CAS Number | 194423-15-9 |
SMILES | C=CC(=O)NC1=CC2=C(C=C1)N=CN=C2NC3=CC(=CC=C3)Br |
Synonyms | PD-168393, PD 168393 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 72 mg/mL (195 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 30% PEG400+0.5% Tween80+5% propylene glycol | 9 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 27.08 mL | 135.42 mL | 270.84 mL |
0.5 mM | 5.42 mL | 27.08 mL | 54.17 mL |
1 mM | 2.71 mL | 13.54 mL | 27.08 mL |
5 mM | 0.54 mL | 2.71 mL | 5.42 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2