Dubermatinib (TP-0903)
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | TP-0903 is a potent and selective Axl kinase inhibitor with IC50 of 27 nM. | ||
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Targets |
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Catalog Num | A15776 |
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Formula | C24H30ClN7O2S |
Molecular Weight | 516.06 |
CAS Number | 1341200-45-0 |
SMILES | CN1CCN(CC1)CC2=CC=C(C=C2)NC3=NC=C(C(=N3)NC4=CC=CC=C4S(=O)(=O)N(C)C)Cl |
Synonyms | TP0903, TP 0903 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | Warmed: 3 mg/mL (5.81 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 1 mg/mL (1.93 mM) | ||
In vivo | 0.5% CMC Na+1% Tween 80 | 28 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 19.38 mL | 96.89 mL | 193.78 mL |
0.5 mM | 3.88 mL | 19.38 mL | 38.76 mL |
1 mM | 1.94 mL | 9.69 mL | 19.38 mL |
5 mM | 0.39 mL | 1.94 mL | 3.88 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2