CPI-203

Catalog No.: A13068
BET bromodomain Inhibitor
CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).
Grouped product items
Product Name Price Stock Qty
CPI-203 5mg
$90.00
In stock
CPI-203 10mg
$170.00
In stock
CPI-203 25mg
$350.00
In stock
CPI-203 50mg
$550.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Adooq's CPI-203 has been cited by 1 publications
  • Derenzini E, .et al. , Cell Rep, 2018, Aug 21;24(8):2155-2166 PMID: 30134175
  • Biological Activity
    Discription CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).
    Product Information
    Catalog Num A13068
    Formula C19H18ClN5OS
    Molecular Weight 399.9
    CAS Number 1446144-04-2
    SMILES CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)N)C4=CC=C(C=C4)Cl)C
    Synonyms CPI203
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro DMSO Warmed: 78 mg/mL (195.04 mM)
    Water Insoluble
    Ethanol 5 mg/mL (12.5 mM)
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 25.01 mL 125.03 mL 250.06 mL
    0.5 mM 5 mL 25.01 mL 50.01 mL
    1 mM 2.5 mL 12.5 mL 25.01 mL
    5 mM 0.5 mL 2.5 mL 5 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

    • Mass

      Concentration

      Volume

      Molecular Weight

    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

    • C1

      V1

      C2

      V2

    • Calculator Reset
    Keywords: buy CPI-203 | CPI-203 Supplier | purchase CPI-203 | CPI-203 cost | CPI-203 manufacturer | order CPI-203 | CPI-203 distributor | buy 1446144-04-2 | 1446144-04-2 Supplier | purchase 1446144-04-2 | 1446144-04-2 cost | 1446144-04-2 manufacturer | order 1446144-04-2 | 1446144-04-2 distributor