G007-LK
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice, | ||
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Targets |
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Catalog Num | A15528 |
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Formula | C25H16ClN7O3S |
Molecular Weight | 529.96 |
CAS Number | 1380672-07-0 |
SMILES | CS(=O)(=O)C1=CN=C(C=C1)C2=NN=C(N2C3=CC=CC=C3Cl)C=CC4=NN=C(O4)C5=CC=C(C=C5)C#N |
Synonyms | G007 LK, G007LK |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 98 mg/mL (184.92 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 18.87 mL | 94.35 mL | 188.69 mL |
0.5 mM | 3.77 mL | 18.87 mL | 37.74 mL |
1 mM | 1.89 mL | 9.43 mL | 18.87 mL |
5 mM | 0.38 mL | 1.89 mL | 3.77 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2