GSK 1210151A (I-BET151)

Catalog No.: A11783
BET Bromodomain Inhibitor
GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
Grouped product items
Product Name Price Stock Qty
GSK 1210151A 5mg
$80.00
In stock
GSK 1210151A 10mg
$120.00
In stock
GSK 1210151A 25mg
$200.00
In stock
GSK 1210151A 50mg
$360.00
In stock
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Important Notice: For research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Adooq's GSK 1210151A (I-BET151) has been cited by 1 publications
  • Momeny M, .et al. , Anticancer Drugs, 2018, Nov;29(10):1011-1020 PMID: 30096128
  • Biological Activity
    Discription GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
    Targets
    Target Value
    Product Information
    Catalog Num A11783
    Formula C23H21N5O3
    Molecular Weight 415.4
    CAS Number 1300031-49-5
    SMILES CC1=C(C(=NO1)C)C2=C(C=C3C(=C2)N=CC4=C3N(C(=O)N4)[C@H](C)C5=CC=CC=N5)OC
    Synonyms GSK1210151A
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro DMSO Insoluble
    Water Insoluble
    Ethanol 27 mg/mL (64.99 mM)
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 24.07 mL 120.37 mL 240.73 mL
    0.5 mM 4.81 mL 24.07 mL 48.15 mL
    1 mM 2.41 mL 12.04 mL 24.07 mL
    5 mM 0.48 mL 2.41 mL 4.81 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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