Itraconazole (Sporanox)

Itraconazole is a relatively potent inhibitor of CYP3A4 with IC50 of 6.1 nM, used as a triazole antifungal agent.
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Product Name Price Stock Qty
Itraconazole (Sporanox) 100mg
$55.00
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Itraconazole (Sporanox) 250mg
$120.00
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Itraconazole (Sporanox) 500mg
$200.00
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Itraconazole (Sporanox) 1000mg
$350.00
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Adooq Products cited in reputable paper
Adooq's Itraconazole (Sporanox) has been cited by 1 publications
  • Paul Mark Medina, .et al. , Transl Oncol, 2021, Jan;14(1):100940 PMID: 33221682
  • Biological Activity
    Discription Itraconazole is a relatively potent inhibitor of CYP3A4 with IC50 of 6.1 nM, used as a triazole antifungal agent.
    Targets
    Target Value
    Product Information
    Catalog Num A10489
    Formula C35H38Cl2N8O4
    Molecular Weight 705.65
    CAS Number 84625-61-6
    SMILES CCC(C)N1C(=O)N(C=N1)C2=CC=C(C=C2)N3CCN(CC3)C4=CC=C(C=C4)OC[C@H]5CO[C@](O5)(CN6C=NC=N6)C7=C(C=C(C=C7)Cl)Cl
    Synonyms Sporanox
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro (25°C) DMSO Warmed: 7 mg/mL (9.91 mM)
    Water Insoluble
    Ethanol Insoluble
    In vivo 5% DMSO+40% PEG 300+10% Tween 80+45% ddH2O 1.66 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 14.17 mL 70.86 mL 141.71 mL
    0.5 mM 2.83 mL 14.17 mL 28.34 mL
    1 mM 1.42 mL 7.09 mL 14.17 mL
    5 mM 0.28 mL 1.42 mL 2.83 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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