A 438079 hydrochloride

Catalog No.: A14983
P2X7 receptor antagonist
A 438079 Hcl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).
Grouped product items
Product Name Price Stock Qty
A 438079 hydrochloride 10mg
$95.00
In stock
A 438079 hydrochloride 25mg
$215.00
In stock
A 438079 hydrochloride 50mg
$395.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Adooq's A 438079 hydrochloride has been cited by 1 publications
  • Zhihua Yi, .et al. , Front Pharmacol, 2018, 9: 593 PMID: 29950989
  • Biological Activity
    Discription A 438079 Hcl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).
    Targets
    Target Value
    Product Information
    Catalog Num A14983
    Formula C13H10Cl3N5
    Molecular Weight 342.61
    CAS Number 899431-18-6
    SMILES C1=CC(=C(C(=C1)Cl)Cl)C2=NN=NN2CC3=CN=CC=C3.Cl
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro (25°C) DMSO 55 mg/mL (160.53 mM)
    Water 55 mg/mL (160.53 mM)
    Ethanol Warmed: 18 mg/mL (52.53 mM)
    In vivo Saline 28 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 29.19 mL 145.94 mL 291.88 mL
    0.5 mM 5.84 mL 29.19 mL 58.38 mL
    1 mM 2.92 mL 14.59 mL 29.19 mL
    5 mM 0.58 mL 2.92 mL 5.84 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

    • Mass

      Concentration

      Volume

      Molecular Weight

    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

    • C1

      V1

      C2

      V2

    • Calculator Reset
    Keywords: buy A 438079 hydrochloride | A 438079 hydrochloride Supplier | purchase A 438079 hydrochloride | A 438079 hydrochloride cost | A 438079 hydrochloride manufacturer | order A 438079 hydrochloride | A 438079 hydrochloride distributor | buy 899431-18-6 | 899431-18-6 Supplier | purchase 899431-18-6 | 899431-18-6 cost | 899431-18-6 manufacturer | order 899431-18-6 | 899431-18-6 distributor