PF 4981517

Catalog No.: A12544
CYP3A4 inhibitor
PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).
Grouped product items
Product Name Price Stock Qty
PF 4981517 5mg
$80.00
In stock
PF 4981517 10mg
$140.00
In stock
PF 4981517 25mg
$280.00
In stock
PF 4981517 50mg
$500.00
In stock
PF 4981517 10mM * 1mL in DMSO
$132.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Biological Activity
Discription PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).
Targets
Target Value
Product Information
Catalog Num A12544
Formula C26H32N8
Molecular Weight 456.59
CAS Number 1390637-82-7
SMILES CC1=CC=C(C=C1)C2=C(C=NN2C)C3=NN(C4=C3C(=NC=N4)N5CC[C@@H](C5)N6CCCCC6)C
Synonyms PF4981517, PF-4981517
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 85 mg/mL (186.16 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.9 mL 109.51 mL 219.01 mL
0.5 mM 4.38 mL 21.9 mL 43.8 mL
1 mM 2.19 mL 10.95 mL 21.9 mL
5 mM 0.44 mL 2.19 mL 4.38 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: buy PF 4981517 | PF 4981517 Supplier | purchase PF 4981517 | PF 4981517 cost | PF 4981517 manufacturer | order PF 4981517 | PF 4981517 distributor | buy 1390637-82-7 | 1390637-82-7 Supplier | purchase 1390637-82-7 | 1390637-82-7 cost | 1390637-82-7 manufacturer | order 1390637-82-7 | 1390637-82-7 distributor