Apabetalone (RVX-208)

Catalog No.: A13956
BET bromodomain inhibitor
RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 uM for BD2, about 170-fold selectivity over BD1.
Grouped product items
Product Name Price Stock Qty
Apabetalone (RVX-208) 10mg
$100.00
In stock
Apabetalone (RVX-208) 25mg
$200.00
In stock
Apabetalone (RVX-208) 50mg
$350.00
In stock
Apabetalone (RVX-208) 10mM * 1mL in DMSO
$75.00
In stock
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Biological Activity
Discription RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 uM for BD2, about 170-fold selectivity over BD1.
Targets
Target Value
Product Information
Catalog Num A13956
Formula C20H22N2O5
Molecular Weight 370.4
CAS Number 1044870-39-4
SMILES CC1=CC(=CC(=C1OCCO)C)C2=NC(=O)C3=C(C=C(C=C3N2)OC)OC
Synonyms RVX-000222
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro (25°C) DMSO 63 mg/mL (170.08 mM)
Water Insoluble
Ethanol Insoluble
In vivo 0.5% CMC Na (1N HCl, PH 2.5-3.0) 7 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27 mL 134.99 mL 269.98 mL
0.5 mM 5.4 mL 27 mL 54 mL
1 mM 2.7 mL 13.5 mL 27 mL
5 mM 0.54 mL 2.7 mL 5.4 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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