Tiplaxtinin (PAI-039)

Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.
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Product Name Price Stock Qty
Tiplaxtinin 5mg
$75.00
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Tiplaxtinin 10mg
$85.00
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Tiplaxtinin 25mg
$200.00
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Adooq Products cited in reputable paper
Adooq's Tiplaxtinin (PAI-039) has been cited by 1 publications
  • Saijo A, .et al. , Cancer Lett, 2018, May 1;421:17-27 PMID: 29448000
  • Biological Activity
    Discription Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.
    Targets
    Target Value
    Product Information
    Catalog Num A14190
    Formula C24H16F3NO4
    Molecular Weight 439.3833
    CAS Number 393105-53-8
    SMILES C1=CC=C(C=C1)CN2C=C(C3=C2C=CC(=C3)C4=CC=C(C=C4)OC(F)(F)F)C(=O)C(=O)O
    Synonyms PAI-039
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro (25°C) DMSO 62 mg/mL (141.1 mM)
    Water Insoluble
    Ethanol Warmed: 15 mg/mL (34.13 mM)
    In vivo 2.0% Tween 80+0.5% methylcellulose 28 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 22.76 mL 113.8 mL 227.59 mL
    0.5 mM 4.55 mL 22.76 mL 45.52 mL
    1 mM 2.28 mL 11.38 mL 22.76 mL
    5 mM 0.46 mL 2.28 mL 4.55 mL
    Useful Calculator

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    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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