TC-E 5001

Catalog No.: A11454
TNKS inhibitor
TC-E 5001 is dual tankyrase (TNKS) inhibitor (Kd values are 79 and 28 nM for TNKS1 and TNKS2 respectively, IC50 = 33 nM for TNKS2) that is devoid of activity at PARP1 and PARP2 (IC50 >19 uM). Inhibits Wnt signaling and stabilizes Axin2 levels.
Grouped product items
Product Name Price Stock Qty
TC-E 5001 5mg
$80.00
In stock
TC-E 5001 10mg
$140.00
In stock
TC-E 5001 50mg
$500.00
In stock
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Biological Activity
Discription TC-E 5001 is dual tankyrase (TNKS) inhibitor (Kd values are 79 and 28 nM for TNKS1 and TNKS2 respectively, IC50 = 33 nM for TNKS2) that is devoid of activity at PARP1 and PARP2 (IC50 >19 uM). Inhibits Wnt signaling and stabilizes Axin2 levels.
Product Information
Catalog Num A11454
Formula C20H19N5O3S
Molecular Weight 409.46
CAS Number 865565-29-3
SMILES CC(N1C(C=C2)=CC=C2OC)=NN=C1SCC3=NC(C(C=C4)=CC=C4OC)=NO3
Synonyms TC-E5001, TC-E-5001
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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