S1RA (E-52862)

Catalog No.: A12504
sigma-1 receptor antagonist
S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ?? 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.
Grouped product items
Product Name Price Stock Qty
S1RA (E-52862) 5mg
$252.00
In stock
S1RA (E-52862) 10mg
$428.00
In stock
S1RA (E-52862) 25mg
$756.00
In stock
S1RA (E-52862) 50mg
$1,260.00
In stock
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Biological Activity
Discription S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ?? 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.
Targets
Target Value
Product Information
Catalog Num A12504
Formula C20H23N3O2
Molecular Weight 337.42
CAS Number 878141-96-9
SMILES CC1=CC(=NN1C2=CC3=CC=CC=C3C=C2)OCCN4CCOCC4
Synonyms E52862, E 52862, MR390; MR 390; MR-390
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 63 mg/mL (186.71 mM)
Water 63 mg/mL (186.71 mM)
Ethanol 18 mg/mL (53.34 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.64 mL 148.18 mL 296.37 mL
0.5 mM 5.93 mL 29.64 mL 59.27 mL
1 mM 2.96 mL 14.82 mL 29.64 mL
5 mM 0.59 mL 2.96 mL 5.93 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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    C2

    V2

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