Canertinib dihydrochloride
Important Notice: For research use only. We do not sell to patients.
Other Forms of Canertinib dihydrochloride
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Important Notice: For research use only. We do not sell to patients.
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Discription | Canertinib dihydrochloride (CI-1033 dihydrochloride) is a potent and irreversible EGFR inhibitor; inhibits cellular EGFR and ErbB2 autophosphorylation with IC50s of 7.4 and 9 nM. | ||
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Catalog Num | A11344 |
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Formula | C24H27Cl3FN5O3 |
Molecular Weight | 558.86 |
CAS Number | 289499-45-2 |
SMILES | C=CC(NC1=CC2=C(N=CN=C2C=C1OCCCN3CCOCC3)NC4=CC=C(C(Cl)=C4)F)=O.[H]Cl.[H]Cl |
Synonyms | CI-1033 dihydrochloride; PD-183805 dihydrochloride |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 88 mg/mL (157.46 mM) | |
Water | 18 mg/mL (32.2 mM) | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 17.89 mL | 89.47 mL | 178.94 mL |
0.5 mM | 3.58 mL | 17.89 mL | 35.79 mL |
1 mM | 1.79 mL | 8.95 mL | 17.89 mL |
5 mM | 0.36 mL | 1.79 mL | 3.58 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2