dBET1

Catalog No.: A16858
BRD4 protein degrader
dBET1 is a potent BRD4 protein degrader based on PROTAC technology with an EC50 of 430 nM.
Grouped product items
Product Name Price Stock Qty
dBET1 2mg
$70.00
In stock
dBET1 5mg
$120.00
In stock
dBET1 10mg
$200.00
In stock
dBET1 50mg
$700.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Biological Activity
Discription dBET1 is a potent BRD4 protein degrader based on PROTAC technology with an EC50 of 430 nM.
Targets
Target Value
Product Information
Catalog Num A16858
Formula C38H37ClN8O7S
Molecular Weight 785.27
CAS Number 1799711-21-9
SMILES O=C(NCCCCNC(COC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)=O)C[C@H]4C5=NN=C(C)N5C6=C(C(C)=C(C)S6)C(C7=CC=C(Cl)C=C7)=N4
Synonyms dBET-1, dBET 1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 89 mg/mL (113.33 mM)
Water <1 mg/mL
Ethanol 35 mg/mL (44.57 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.73 mL 63.67 mL 127.34 mL
0.5 mM 2.55 mL 12.73 mL 25.47 mL
1 mM 1.27 mL 6.37 mL 12.73 mL
5 mM 0.25 mL 1.27 mL 2.55 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: buy dBET1 | dBET1 Supplier | purchase dBET1 | dBET1 cost | dBET1 manufacturer | order dBET1 | dBET1 distributor | buy 1799711-21-9 | 1799711-21-9 Supplier | purchase 1799711-21-9 | 1799711-21-9 cost | 1799711-21-9 manufacturer | order 1799711-21-9 | 1799711-21-9 distributor