dBET1
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | dBET1 is a potent BRD4 protein degrader based on PROTAC technology with an EC50 of 430 nM. | ||
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Targets |
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Catalog Num | A16858 |
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Formula | C38H37ClN8O7S |
Molecular Weight | 785.27 |
CAS Number | 1799711-21-9 |
SMILES | O=C(NCCCCNC(COC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)=O)C[C@H]4C5=NN=C(C)N5C6=C(C(C)=C(C)S6)C(C7=CC=C(Cl)C=C7)=N4 |
Synonyms | dBET-1, dBET 1 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 89 mg/mL (113.33 mM) | |
Water | <1 mg/mL | ||
Ethanol | 35 mg/mL (44.57 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 12.73 mL | 63.67 mL | 127.34 mL |
0.5 mM | 2.55 mL | 12.73 mL | 25.47 mL |
1 mM | 1.27 mL | 6.37 mL | 12.73 mL |
5 mM | 0.25 mL | 1.27 mL | 2.55 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2