Eptapirone (F-11440)

Catalog No.: A18338
5-HT1A receptor agonist
Eptapirone is a potent, selective, high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential. The affinity of F 11440 for 5-HT1A binding sites (pKi, 8.33) was higher than that of buspirone (pKi, 7.50), and somewhat lower than that of flesinoxan (pKi, 8.91). In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone.
Grouped product items
Product Name Price Stock Qty
Eptapirone (F-11440) 1mg
$40.00
In stock
Eptapirone (F-11440) 5mg
$100.00
In stock
Eptapirone (F-11440) 10mg
$180.00
In stock
Eptapirone (F-11440) 50mg
$560.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Biological Activity
Discription Eptapirone is a potent, selective, high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential. The affinity of F 11440 for 5-HT1A binding sites (pKi, 8.33) was higher than that of buspirone (pKi, 7.50), and somewhat lower than that of flesinoxan (pKi, 8.91). In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone.
Targets
Target Value
Product Information
Catalog Num A18338
Formula C16H23N7O2
Molecular Weight 345.407
CAS Number 179756-58-2
SMILES O=C(N1C)N(CCCCN2CCN(C3=NC=CC=N3)CC2)N=CC1=O
Synonyms F11440, F 11440
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: buy Eptapirone (F-11440) | Eptapirone (F-11440) Supplier | purchase Eptapirone (F-11440) | Eptapirone (F-11440) cost | Eptapirone (F-11440) manufacturer | order Eptapirone (F-11440) | Eptapirone (F-11440) distributor | buy 179756-58-2 | 179756-58-2 Supplier | purchase 179756-58-2 | 179756-58-2 cost | 179756-58-2 manufacturer | order 179756-58-2 | 179756-58-2 distributor