GSK5182

Catalog No.: A19383
ERRγ agonist
GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα.
Grouped product items
Product Name Price Stock Qty
GSK5182 1mg
$80.00
In stock
GSK5182 5mg
$250.00
In stock
GSK5182 10mg
$410.00
In stock
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Important Notice: For research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Adooq's GSK5182 has been cited by 1 publications
  • Sen He, .et al. , Toxicology, 2021, May 4;457:152805 PMID: 33961950
  • Biological Activity
    Discription GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα.
    Targets
    Target Value
    Product Information
    Catalog Num A19383
    Formula C27H31NO3
    Molecular Weight 417.54
    CAS Number 877387-37-6
    SMILES OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3
    Synonyms GSK 5182, GSK-5182
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro DMSO 78 mg/mL
    Water Insoluble
    Ethanol 78 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 23.95 mL 119.75 mL 239.5 mL
    0.5 mM 4.79 mL 23.95 mL 47.9 mL
    1 mM 2.39 mL 11.97 mL 23.95 mL
    5 mM 0.48 mL 2.39 mL 4.79 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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